Liquid-phase synthesis of 2,3-dihydro-4-pyridones: one-pot three-component aza Diels-Alder reaction of Danishefsky's diene with aldehydes and PEG-supported amine

被引：13

作者：

Guo, HC ^{[1
]}

Ding, KL ^{[1
]}

机构：

[1] Chinese Acad Sci, Shanghai Inst Organ Chem, State Key Lab Organomet Chem, Shanghai 200032, Peoples R China

来源：

TETRAHEDRON LETTERS | 2003年 / 44卷 / 37期

基金：

中国国家自然科学基金;

关键词：

D O I：

10.1016/S0040-4039(03)01708-8

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

An efficient liquid-phase synthesis technique for the construction of 2,3-dihydro-4-pyridones on soluble polymer support has been developed, which utilized one-pot reaction of Danishefsky's diene with aldehydes and polymer-supported amine. (C) 2003 Elsevier Ltd. All rights reserved.

引用

页码：7103 / 7106

页数：4

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