Drug metabolism and pharmacokinetic strategies for oligonucleotide- and mRNA-based drug development

被引:45
作者
Andersson, Shalini [1 ]
Antonsson, Madeleine [1 ]
Elebring, Marie [1 ]
Jansson-Lofmark, Rasmus [1 ]
Weidolf, Lars [1 ]
机构
[1] AstraZeneca Gothenburg, Innovat Med Biotech Unit, Drug Metab & Pharmacokinet, Cardiovasc Renal & Metab, SE-43183 Molndal, Sweden
关键词
2ND-GENERATION ANTISENSE OLIGONUCLEOTIDE; TARGETING APOLIPOPROTEIN B-100; N-ACETYL GALACTOSAMINE; KINASE-C-ALPHA; THERAPEUTIC OLIGONUCLEOTIDES; PHOSPHOROTHIOATE OLIGONUCLEOTIDE; MASS-SPECTROMETRY; ADVANCED CANCER; RAT-LIVER; PHASE-I;
D O I
10.1016/j.drudis.2018.05.030
中图分类号
R9 [药学];
学科分类号
1007 ;
摘要
Oligonucleotide and modified mRNA therapeutics have great potential to treat diseases that are currently challenging to cure and are expanding into global and chronic disease areas such as cancer and various cardiovascular diseases. Advanced drug delivery systems or ligand-drug conjugates are utilized to achieve 'the right dose to the right target' to benefit efficacy and safety in patients. Chemistry and ADME characteristics distinguish these therapeutics from small molecules. Understanding the scalability and translatability between species and compound properties is crucial for robust nonclinical PKPD predictions to support clinical study design. Although the field has been developing for three decades, there is still room for innovation but also a need for nonclinical regulatory guidance to address these new modalities.
引用
收藏
页码:1733 / 1745
页数:13
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