共 30 条
Morroniside protects against cerebral ischemia/reperfusion injury by inhibiting neuron apoptosis and MMP2/9 expression
被引:44
作者:

Zeng, Guoyong
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机构:
Nanchang Univ, Affiliated Ganzhou Hosp, Dept Neurol, Ganzhou 341000, Jiangxi, Peoples R China Nanchang Univ, Affiliated Ganzhou Hosp, Dept Neurol, Ganzhou 341000, Jiangxi, Peoples R China

Ding, Weijiang
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机构:
Nanchang Univ, Affiliated Hosp 2, Dept Neurol, 1 Minde Rd, Nanchang 330006, Jiangxi, Peoples R China Nanchang Univ, Affiliated Ganzhou Hosp, Dept Neurol, Ganzhou 341000, Jiangxi, Peoples R China

Li, Yin
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h-index: 0
机构:
Nanchang Univ, Affiliated Hosp 2, Dept Neurol, 1 Minde Rd, Nanchang 330006, Jiangxi, Peoples R China Nanchang Univ, Affiliated Ganzhou Hosp, Dept Neurol, Ganzhou 341000, Jiangxi, Peoples R China

Sun, Meiying
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h-index: 0
机构:
Peoples Hosp Fuzhou, Dept Neurol, Fuzhou 344000, Jiangxi, Peoples R China Nanchang Univ, Affiliated Ganzhou Hosp, Dept Neurol, Ganzhou 341000, Jiangxi, Peoples R China

Deng, Liying
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h-index: 0
机构:
Nanchang Univ, Affiliated Hosp 2, Dept Neurol, 1 Minde Rd, Nanchang 330006, Jiangxi, Peoples R China Nanchang Univ, Affiliated Ganzhou Hosp, Dept Neurol, Ganzhou 341000, Jiangxi, Peoples R China
机构:
[1] Nanchang Univ, Affiliated Ganzhou Hosp, Dept Neurol, Ganzhou 341000, Jiangxi, Peoples R China
[2] Nanchang Univ, Affiliated Hosp 2, Dept Neurol, 1 Minde Rd, Nanchang 330006, Jiangxi, Peoples R China
[3] Peoples Hosp Fuzhou, Dept Neurol, Fuzhou 344000, Jiangxi, Peoples R China
关键词:
morroniside;
cerebral ischemia;
reperfusion injury;
matrix metalloproteinase-2;
matrix metalloproteinase-9;
ISCHEMIA-REPERFUSION INJURY;
BLOOD-BRAIN-BARRIER;
CORNI FRUCTUS;
UP-REGULATION;
RATS;
MATRIX;
CELLS;
CONTRIBUTES;
DISRUPTION;
ACTIVATION;
D O I:
10.3892/etm.2018.6457
中图分类号:
R-3 [医学研究方法];
R3 [基础医学];
学科分类号:
1001 ;
摘要:
The aim of the present study was to investigate the effect of morroniside against matrix metalloproteinase (MMP)2/9 and focal cerebral ischemia/reperfusion (I/R) injury in rats. A rat model of focal cerebral I/R injury rats was established and rats were administered with 30, 90 or 270 mg/kg/day morroniside for 7 days. The expression of MMP2/9 and neuronal apoptosis were assessed. In addition, the expression of active caspase-3, B-cell lymphoma 2 (Bcl-2) and Bcl-2-associated X protein (Bax) were measured. The results revealed that MMP2 and MMP9 expression was upregulated and the percentage of apoptotic neurons was increased in rats with focal cerebral I/R injury compared with the control. However, treatment with morroniside significantly inhibited I/R-induced MMP2/9 expression and neuron apoptosis compared with the untreated I/R injury group. Morroniside administration also decreased the expression of active caspase-3 and increased the Bcl-2/Bax ratio compared with untreated rats with focal cerebral I/R injury. The inhibitory effect of morroniside on MMP2/9 expression and neuron apoptosis was dose dependent. In summary, the results of the present study suggest that morroniside is able to protect against cerebral I/R injury in the brain and may have potential as a therapeutic treatment for patients who have suffered a stroke.
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页码:2229 / 2234
页数:6
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Guangxi Med Univ, Affiliated Hosp 1, Western Hosp, Dept Emergency, Nanning 530021, Peoples R China Guangxi Med Univ, Affiliated Hosp 1, Western Hosp, Dept Emergency, Nanning 530021, Peoples R China

Li, Chaoqian
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Guangxi Med Univ, Affiliated Hosp 1, Western Hosp, Dept Emergency, Nanning 530021, Peoples R China Guangxi Med Univ, Affiliated Hosp 1, Western Hosp, Dept Emergency, Nanning 530021, Peoples R China
[10]
MMP-2 siRNA PROTECTS AGAINST CONTRACTILE DYSFUNCTION IN CARDIOMYOCYTES SUBJECTED TO ISCHEMIA/REPERFUSION
[J].
Lin, H.
;
Sra, B.
;
Cadete, V. J.
;
Sawicka, J.
;
Cayabyab, F. S.
;
Sawicki, G.
.
CANADIAN JOURNAL OF CARDIOLOGY,
2012, 28 (05)
:S396-S397

Lin, H.
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Sra, B.
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Cadete, V. J.
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Sawicka, J.
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Cayabyab, F. S.
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Sawicki, G.
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