A convenient modified synthesis of 5-pyridinyl-1,3,4-thiadiazole-2-carboxamides

被引:5
作者
Myannik, K. A. [1 ]
Yarovenko, V. N. [1 ]
Rodionova, G. M. [2 ]
Baryshnikova, T. K. [1 ]
Krayushkin, M. M. [1 ]
机构
[1] Russian Acad Sci, ND Zelinsky Inst Organ Chem, Moscow 119991, Russia
[2] IM Sechenov First Moscow State Med Univ, Moscow 119991, Russia
基金
俄罗斯科学基金会;
关键词
Pyridine carboxaldehydes; 1,3,4-thiadiazoles; oxamic acid thiohydrazides; pyridinyl thiadiazoles; carboxamides; THIOHYDRAZIDES;
D O I
10.24820/ark.5550190.p010.233
中图分类号
O62 [有机化学];
学科分类号
070303 ; 081704 ;
摘要
A general one-pot procedure is developed for the synthesis of 5-pyridinyl-1,3,4-thiadiazole-2-carboxamides by the reaction of pyridine carboxaldehydes with oxamic acid thiohydrazides.
引用
收藏
页码:316 / 325
页数:10
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