Discovery of clinical candidate BMS-986115, an oral pan-Notch inhibitor for the treatment of cancer

被引:0
作者
Gavai, Ashvinikumar V. [1 ]
Delucca, George [1 ]
Norris, Derek [1 ]
O'Malley, Daniel [1 ]
Zhao, Yufen [1 ]
Fink, Brian [1 ]
Quesnelle, Claude [1 ]
Han, Wen-Ching [1 ]
Gill, Patrice [1 ]
Vaccaro, Wayne [1 ]
Tram Huynh [1 ]
Ahuja, Vijay [1 ]
Saulnier, Mark [1 ]
Frennesson, David [1 ]
Tebben, Andrew [3 ]
Rampulla, Richard [6 ]
Wu, Dauh-Rurng [6 ]
Wang, Chunlei [4 ]
Zhang, Yingru [4 ]
Mathur, Arvind [6 ]
Wang, Haiqing [4 ]
Moore, Robin [4 ]
Yang, Zheng [4 ]
Ranasinghe, Asoka [4 ]
Tye, Ching Kim [4 ]
Su, Ching [4 ]
Everlof, Gerry [4 ]
Ruan, Qian [4 ]
Yarde, Melissa [5 ]
Menard, Krista [2 ]
Wen, Mei-Li [2 ]
Hunt, John [2 ]
Vite, Gregory [1 ]
Westhouse, Richard [4 ]
Lee, Francis [2 ]
机构
[1] Bristol Myers Squibb R&D, Dept Oncol Chem, Princeton, NJ 08543 USA
[2] Bristol Myers Squibb R&D, Dept Oncol, Princeton, NJ 08543 USA
[3] Bristol Myers Squibb R&D, Dept Comp Assisted Drug Design, Princeton, NJ 08543 USA
[4] Bristol Myers Squibb R&D, Dept Pharmaceut Candidate Optimizat, Princeton, NJ 08543 USA
[5] Bristol Myers Squibb R&D, Dept Leads Discovery & Optimizat, Princeton, NJ 08543 USA
[6] Bristol Myers Squibb R&D, Dept Discovery Synth, Princeton, NJ 08543 USA
来源
ABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY | 2014年 / 248卷
关键词
D O I
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中图分类号
O6 [化学];
学科分类号
0703 ;
摘要
350-MEDI
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页数:1
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