An Efficient Synthesis of trans-N-{2-[4-(2-Methoxyphenyl)piperazinyl]ethyl}-N-(2-pyridy1)-N-(4-tosyloxymethylcyclohexane)carboxamide, A Precursor of [18F]Mefway for Imaging 5-HT1A Receptor

被引：3

作者：

Choi, Jae Yong ^{[1
,2
]}

Kim, Chul Hoon ^{[2
]}

Kim, Jung Young ^{[3
,4
,5
]}

Ha, Hyun-Joon ^{[4
,5
]}

Ryu, Young Hoon ^{[1
]}

机构：

[1] Yonsei Univ, Coll Med, Gangnam Severance Hosp, Dept Nucl Med, Seoul 135720, South Korea

[2] Yonsei Univ, Coll Med, Dept Pharmacol, Brain Res Inst,Brain Korea Project Med Sci 21, Seoul 120752, South Korea

[3] Korea Inst Radiol & Med Sci, Mol Imaging Res Ctr, Seoul 139706, South Korea

[4] Hankuk Univ Foreign Studies, Dept Chem, Yongin 449791, Kyunggi Do, South Korea

[5] Hankuk Univ Foreign Studies, Prot Res Ctr Bioind, Yongin 449791, Kyunggi Do, South Korea

来源：

BULLETIN OF THE KOREAN CHEMICAL SOCIETY | 2010年 / 31卷 / 08期

关键词：

Serotonin receptors; 5-HT1A; F-18]Mefway; WAY-100635; IN-VIVO; PET; ANTAGONISTS; WAY-100635; RADIOLIGANDS; ANALOGS;

D O I：

10.5012/bkcs.2010.31.8.2371

中图分类号：

O6 [化学];

学科分类号：

0703 ;

摘要：

[No abstract available]

引用

页码：2371 / 2374

页数：4

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