Diversity-orientated synthesis of 3,5-bis(arylamino)pyrazoles

被引：13

作者：

Degorce, Sebastien ^{[1
]}

Jung, Frederic H. ^{[1
]}

Harris, Craig S. ^{[1
]}

Koza, Patrice ^{[1
]}

Lecoq, Jonathan ^{[1
]}

Stevenin, Arnaud ^{[1
]}

机构：

[1] AstraZeneca, Oncol iMed, Ctr Rech, ZI Pompelle, F-51689 Reims 2, France

来源：

TETRAHEDRON LETTERS | 2011年 / 52卷 / 50期

关键词：

ISOTHIOCYANATE; DERIVATIVES;

D O I：

10.1016/j.tetlet.2011.09.150

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

The synthesis of differentially-substituted 3,5-bis(arylamino)pyrazoles has not yet been documented. During our investigation, we managed to develop a novel, entirely combinatorial synthesis of 3,5-bis(arylamino)pyrazoles relying on a simple one-pot two-step operation. (C) 2011 Elsevier Ltd. All rights reserved.

引用

页码：6719 / 6722

页数：4

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