An efficient one-pot synthesis of 3-substituted-5-amino1,2,4-thiadiazoles from isothiocyanates and amidines

被引:21
|
作者
Wu, Yong-Jin [1 ]
Zhang, Yunhui [1 ]
机构
[1] Bristol Myers Squibb Res & Dev, Dept Neurosci Chem, Wallingford, CT 06492 USA
关键词
D O I
10.1016/j.tetlet.2008.03.030
中图分类号
O62 [有机化学];
学科分类号
070303 ; 081704 ;
摘要
An efficient one-pot synthesis of 3-substituted-5-amino-1,2,4-thiadiazoles from isothiocyanates and amidines is described. (c) 2008 Elsevier Ltd. All rights reserved.
引用
收藏
页码:2869 / 2871
页数:3
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