Synthesis of [1,2,3]triazolo[4,5-d]pyrimidine 3-oxides

被引：6

作者：

Yavolovskii, AA ^{[1
]}

Ivanov, EI ^{[1
]}

Mazepa, AV ^{[1
]}

Ivanov, YE ^{[1
]}

机构：

[1] Natl Acad Sci Ukraine, Bogatskii Physicochem Inst, Odessa, Ukraine

来源：

RUSSIAN JOURNAL OF GENERAL CHEMISTRY | 2003年 / 73卷 / 09期

关键词：

Pyrimidine; Hydroxyamino; Benzenediazonium; Benzenediazonium Salt;

D O I：

10.1023/B:RUGC.0000016004.71832.bb

中图分类号：

O6 [化学];

学科分类号：

0703 ;

摘要：

[1,2,3]Triazolo[4,5-d]pyrimidine 3-oxides were synthesized by replacement of the amino group in 6-aminouracil by hydroxyamino, coupling of the resulting 6-hydroxyaminopyrimidine with benzenediazonium salts, and oxidation of 6-hydroxyamino-5-phenylazouracils with a solution of K-3[Fe(CN)(6)] in water.

引用

页码：1486 / 1488

页数：3

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