A facile microwave-assisted synthesis of 8,9-cycloalkathieno[3,2-e] [1,2,4]triazolo[1,5-c]pyrimidin-5(6H)-ones

被引：3

作者：

Kaur, Rajwinder ^{[1
,2
]}

Kishore, D. Pran ^{[1
,2
]}

Narayana, B. Lakshmi ^{[1
,2
]}

Rao, K. Venkat ^{[1
,2
]}

Balakumar, C. ^{[3
]}

Rajkumar, V. ^{[4
,5
]}

Rao, A. Raghuram ^{[1
,2
]}

机构：

[1] Panjab Univ, Univ Inst Pharmaceut Sci, Pharmaceut Chem Div, Chandigarh 160014, India

[2] Panjab Univ, Ctr Adv Study Pharmaceut Sci UGC CAS, Chandigarh 160014, India

[3] Panjab Univ, CPEBS, Chandigarh 160014, India

[4] Panjab Univ, Dept Chem, Chandigarh 160014, India

[5] Panjab Univ, Ctr Adv Study Chem UGC CAS, Chandigarh 160014, India

来源：

JOURNAL OF CHEMICAL SCIENCES | 2011年 / 123卷 / 01期

关键词：

Microwave-irradiation; pyrimidinones; 1,2,4-triazole; aryl hydrazides; condensation; ADENOSINE RECEPTOR ANTAGONISTS; A(2A); POTENT; TRIAZOLOTHIENOPYRIMIDINES; PHARMACOLOGY; NONXANTHINE; DERIVATIVES;

D O I：

10.1007/s12039-011-0067-6

中图分类号：

O6 [化学];

学科分类号：

0703 ;

摘要：

A new series of fused thieno[3,2-e][1,2,4]triazolo[1,5-c]pyrimidinones was synthesized by condensation of ethyl-3-cyano-4,5,6,7-tetrahydrobenzo[b]thiophene-2-yl carbamate with aryl acid hydrazides in quantitative yields using a facile, one-pot procedure under microwave-assisted conditions.

引用

页码：69 / 73

页数：5

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