1,3,4-oxa(thia)diazino [i,j]-annelated quinolines: a new type of key intermediate in the synthesis of tricyclic fluoroquinolones

被引:0
作者
Lipunova, GN [1 ]
Nosova, EV [1 ]
Charushin, VN [1 ]
Sidorova, LP [1 ]
Chasovskikh, OM [1 ]
机构
[1] Urals State Tech Univ, Dept Organ Chem, Ekaterinburg 620002, Russia
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D O I
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中图分类号
O6 [化学];
学科分类号
0703 ;
摘要
The synthesis of new derivatives of 1,3,4-oxa(thia)diazino[6,5,4-i,j]-quinolines, which have a structure that is very similar to the ofloxacin skeleton, by intramolecular cyclizations of ethyl 3-(R-carbonylhydrazino)- and 3- (R-thiocarbonylhydrazino)-substituted 2-polyfluorobenzoyl acrylates, is described.
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页码:131 / 133
页数:3
相关论文
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