Syntheses of 1-substituted-3-aminopyrazoles

被引:14
作者
Ji, Nan [1 ]
Meredith, Erik [1 ]
Liu, Donglei [1 ]
Adams, Christopher M. [1 ]
Artman, Gerald D., III [1 ]
Jendza, Keith C. [1 ]
Ma, Fupeng [1 ]
Mainolfi, Nello [1 ]
Powers, James J. [1 ]
Zhang, Chun [1 ]
机构
[1] Novartis Inst BioMed Res, Cambridge, MA 02139 USA
关键词
CUPRIC ACETATE; ACID;
D O I
10.1016/j.tetlet.2010.10.073
中图分类号
O62 [有机化学];
学科分类号
070303 ; 081704 ;
摘要
A series of 1-substituted-3-aminopyrazoles were prepared via Chan-Lam coupling reactions, alkylation, and pyrazole ring formation. (C) 2010 Elsevier Ltd. All rights reserved.
引用
收藏
页码:6799 / 6801
页数:3
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