An efficient one-pot synthesis of 2-hydroxyalkyl dithiocarbamates

被引：24

作者：

Cui, JL ^{[1
]}

Ge, ZM ^{[1
]}

Cheng, TM ^{[1
]}

Li, RT ^{[1
]}

机构：

[1] Peking Univ, Sch Pharmaceut Sci, Dept Biol Chem, Beijing 100083, Haidian Dist, Peoples R China

来源：

SYNTHETIC COMMUNICATIONS | 2003年 / 33卷 / 12期

基金：

中国国家自然科学基金;

关键词：

2-hydroxyalkyl dithiocarbamate; ring opening of epoxide; regioselective reaction; anhydrous potassium phosphate; carbon disulfide;

D O I：

10.1081/SCC-120021023

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

In the presence of anhydrous potassium phosphate, epoxides reacted with carbon disulfide and primary or secondary amines in acetone to give the corresponding 2-hydroxyalkyl dithiocarbamates regioselectively in moderate to good yield.

引用

页码：1969 / 1976

页数：8

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