Development of a Vaccinia H1-Related (VHR) Phosphatase Inhibitor with a Nonacidic Phosphate-Mimicking Core Structure

被引：19
作者：
Hirai, Go [1 ]
Tsuchiya, Ayako [1 ]
Koyama, Yusuke [1 ]
Otani, Yuko [1 ]
Oonuma, Kana [1 ]
Dodo, Kosuke [1 ,2 ]
Simizu, Siro [1 ]
Osada, Hiroyuki [1 ]
Sodeoka, Mikiko [1 ,2 ]
机构：
[1] RIKEN Adv Sci Inst, Wako, Saitama 3510198, Japan
[2] ERATO Japan Sci & Technol Agcy, Sodeoka Live Cell Chem Project, Wako, Saitama 3510198, Japan
来源：
CHEMMEDCHEM | 2011年 / 6卷 / 04期
关键词：
cell cycle; dual-specificity protein phosphatases; enzymes; inhibitors; natural product analogues; PROTEIN-TYROSINE PHOSPHATASES; DUAL-SPECIFICITY PHOSPHATASES; TENUAZONIC ACID ANALOGS; CELL-CYCLE ARREST; TETRONIC ACID; HIV-1; PROTEASE; TETRAMIC ACID; ERK; PHOSPHORYLATION; LIBRARY;
D O I：
10.1002/cmdc.201100107
中图分类号：
R914 [药物化学];
学科分类号：
100701 ;
摘要：
[No abstract available]
引用
收藏
页码：617 / 622
页数：6
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