(Bromodimethyl)sulfonium bromide:: an inexpensive reagent for the solvent-free, one-pot synthesis of α-aminophosphonates

被引：70

作者：

Kudrimoti, S ^{[1
]}

Bommena, VR ^{[1
]}

机构：

[1] Indian Inst Chem Technol, Div Organ 2, Hyderabad 500007, Andhra Pradesh, India

来源：

TETRAHEDRON LETTERS | 2005年 / 46卷 / 07期

关键词：

alpha-aminophosphonates; (bromodimethyl)sulfonium; bromide; imine;

D O I：

10.1016/j.tetlet.2004.12.070

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

A novel solvent-free, one-pot synthesis of alpha-aminophosphonates in the presence of catalytic (bromodimethyl)sulfonium bromide at room temperature in high yields is reported. (C) 2004 Elsevier Ltd. All rights reserved.

引用

页码：1209 / 1210

页数：2

共 28 条

[1]

[Anonymous], ROLE PHOSPHONATES LI

[2] SYNTHESIS AND STRUCTURE-ACTIVITY-RELATIONSHIPS OF ANTIBACTERIAL PHOSPHONOPEPTIDES INCORPORATING (1-AMINOETHYL)PHOSPHONIC ACID AND (AMINOMETHYL)PHOSPHONIC ACID [J].

ATHERTON, FR ;

HASSALL, CH ;

LAMBERT, RW .

JOURNAL OF MEDICINAL CHEMISTRY, 1986, 29 (01) :29-40

[3] 1-AMINOALKYLPHOSPHONOUS ACIDS .1. ISOSTERES OF THE PROTEIN AMINO-ACIDS [J].

BAYLIS, EK ;

CAMPBELL, CD ;

DINGWALL, JG .

JOURNAL OF THE CHEMICAL SOCIETY-PERKIN TRANSACTIONS 1, 1984, (12) :2845-2853

[4]

BRUKE TR, 1994, BIOCHEM BIOPH RES CO, V204, P129

[5]

BRUKE TR, 1995, J MED CHEM, V38, P1386

[6] THE SYNTHESIS OF ESTERS OF SUBSTITUTED AMINO PHOSPHONIC ACIDS [J].

FIELDS, EK .

JOURNAL OF THE AMERICAN CHEMICAL SOCIETY, 1952, 74 (06) :1528-1531

[7]

GANCARZ R, 1977, SYNTHESIS-STUTTGART, P625

[8] PHOSPHORUS AMINO-ACID-ANALOGS AS INHIBITORS OF LEUCINE AMINOPEPTIDASE [J].

GIANNOUSIS, PP ;

BARTLETT, PA .

JOURNAL OF MEDICINAL CHEMISTRY, 1987, 30 (09) :1603-1609

[9]

Kabachnik M. I., 1954, IZV AKAD NAUK K, P1024

[10]

KABACHNIK MI, 1953, B ACAD SCI USSR CH+, P1126

← 1 2 3 →