Synthesis of 2-azetidinones bearing benzothiazole moiety as possible antibacterials

被引：0
|
作者：
Ojha, KG [1 ]
Jaisinghani, N [1 ]
Tahiliani, H [1 ]
机构：
[1] MDS Univ, Dept Appl Chem, Ajmer 305009, India
来源：
ASIAN JOURNAL OF CHEMISTRY | 2001年 / 13卷 / 02期
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中图分类号：
O6 [化学];
学科分类号：
0703 ;
摘要：
Benzothiazolyl derivatives of 2-azetidinones (III) were synthesised by the condensation of aromatic aldehydes with various substituted 2-aminobenzothiazoles (I). The condensed products (II) were treated with acetyl chloride in presence of triethylamine in dioxane to get title compounds (III). These compounds were screened for their antibacterial activities against S, aureus. Pseudomonas klebsiella, Proteus mirabilis and E. coli.
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页码：798 / 800
页数：3
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