Crystal structure of (E)-N'-((4-aminophenyl)sulfonyl)-N,N-dimethylformimidamide, C9H13N3O2S

被引:0
作者
Abdel-Aziz, Alaa A-M [1 ]
El-Azab, Adel S. [1 ]
Ghabbour, Hazem A. [2 ]
Obaidullaha, Ahmad J. [1 ]
机构
[1] King Saud Univ, Coll Pharm, Dept Pharmaceut Chem, POB 2457, Riyadh 11451, Saudi Arabia
[2] Univ Mansoura, Fac Pharm, Dept Med Chem, Mansoura 35516, Egypt
来源
ZEITSCHRIFT FUR KRISTALLOGRAPHIE-NEW CRYSTAL STRUCTURES | 2020年 / 235卷 / 02期
关键词
SULFONAMIDES; DERIVATIVES;
D O I
10.1515/ncrs-2019-0781
中图分类号
O7 [晶体学];
学科分类号
0702 ; 070205 ; 0703 ; 080501 ;
摘要
C9H13N3O2S, monoclinic, P2(1)/c (no. 14), a = 8.0984(4) angstrom, b = 17.3203(10) angstrom, c = 9.6802(4) angstrom, beta = 124.031(3)degrees, V = 1125.26(10) angstrom(3), Z = 4, R-gt(F) = 0.0504, wR(ref)(F-2) = 0.1275, T = 293(2) K.
引用
收藏
页码:483 / 484
页数:2
相关论文
共 11 条
[1]   Synthesis and anti-inflammatory activity of sulfonamides and carboxylates incorporating trimellitimides: Dual cyclooxygenase/carbonic anhydrase inhibitory actions [J].
Abdel-Aziz, Alaa A. -M. ;
Angeli, Andrea ;
El-Azab, Adel S. ;
Hammouda, Mohammed E. A. ;
El-Sherbeny, Magda A. ;
Supuran, Claudiu T. .
BIOORGANIC CHEMISTRY, 2019, 84 :260-268
[2]   Carbonic anhydrase inhibitory activity of sulfonamides and carboxylic acids incorporating cyclic imide scaffolds [J].
Abdel-Aziz, Alaa A. -M. ;
El-Azab, Adel S. ;
Ceruso, Mariangela ;
Supuran, Claudiu T. .
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2014, 24 (22) :5185-5189
[3]   Investigation of arenesulfonyl-2-imidazolidinones as potent carbonic anhydrase inhibitors [J].
Abdel-Aziz, Alaa A-M. ;
El-Azab, Adel S. ;
Ekinci, Deniz ;
Senturk, Murat ;
Supuran, Claudiu T. .
JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY, 2015, 30 (01) :81-84
[4]   Design, synthesis, single-crystal and preliminary antitumor activity of novel arenesulfonylimidazolidin-2-ones [J].
Abdel-Aziz, Alaa A-M. ;
El-Azab, Adel S. ;
El-Subbagh, Hussein I. ;
Al-Obaid, Abdulrahman M. ;
Alanazi, Amer M. ;
Al-Omar, Mohamed A. .
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2012, 22 (05) :2008-2014
[5]   Structure-based design of phthalimide derivatives as potential cyclooxygenase-2 (COX-2) inhibitors: Anti-inflammatory and analgesic activities [J].
Alanazi, Amer M. ;
El-Azab, Adel S. ;
Al-Suwaidan, Ibrahim A. ;
ElTahir, Kamal Eldin H. ;
Asiri, Yousif A. ;
Abdel-Aziz, Naglaa I. ;
Abdel-Aziz, Alaa A. -M. .
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2015, 92 :115-123
[6]  
Bruker, 2014, BRUKER APEX S SADABS
[7]   Inhibition of carbonic anhydrase isoforms I, II, IV, VII and XII with carboxylates and sulfonamides incorporating phthalimide/phthalic anhydride scaffolds [J].
El-Azab, Adel S. ;
Abdel-Aziz, Alaa A. -M. ;
Ayyad, Rezk R. ;
Ceruso, Mariangela ;
Supuran, Claudiu T. .
BIOORGANIC & MEDICINAL CHEMISTRY, 2016, 24 (01) :20-25
[8]   Improved synthesis of N-sulfonylformamidine derivatives promoted by thionyl chloride [J].
Hudabaierdi, Ruzeahong ;
Wusiman, Abudureheman ;
Mulati, Ayinigeer .
PHOSPHORUS SULFUR AND SILICON AND THE RELATED ELEMENTS, 2017, 192 (05) :485-489
[9]  
Sheldrick GM, 2015, ACTA CRYSTALLOGR C, V71, P3, DOI [10.1107/S2053273314026370, 10.1107/S2053229614024218, 10.1107/S0108767307043930]
[10]   A simple preparation of N,N-dimethyl-N′-alkyl (aryl) sulfonylformamidines [J].
Silva, AL ;
Covarrubias-Zúñiga, A ;
Maldonado, LA .
ORGANIC PREPARATIONS AND PROCEDURES INTERNATIONAL, 2002, 34 (05) :545-549