Synthesis of new (4-acetonylidene-2,6,8,9-tetramethyl-7H-imidazo[1,5,4-e,f][1,5]benzodiazepine) derivatives

被引：2

作者：

El Kihel, Abdellatif ^{[1
]}

Ahbala, Mustapha ^{[1
]}

Mouzdahir, Abdelkrim ^{[1
]}

Snader, Naima ^{[1
]}

Essassi, El Mokhtar ^{[2
]}

Bauchat, Patrick ^{[3
]}

Danion-Bougot, Renee ^{[3
]}

机构：

[1] Chim Bioorgan Lab, Fac Sci, El Jadida 24000, Morocco

[2] Assoc CNCPRST, Fac Sci, Lab Chim Organ Heterocycl, Rabat, Maroc, Morocco

[3] Univ Rennes 1, Rennes, France

来源：

SYNTHETIC COMMUNICATIONS | 2008年 / 38卷 / 02期

关键词：

acetylacetone; 7-amino-2,5,6-trimethylbenzimidazole; ethyl acetoacetate; imidazo[1,5,4-e,f][1,5]benzodiazepine;

D O I：

10.1080/00397910701738933

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

Imidazobenzodiazepine derivatives were obtained by cyclization of the condensation products 7-amino-2,5,6-trimethylbenzimidazole with acetylacetone and ethyl acetoacetate. By careful examination of spectroscopic data and the open-chain intermediate isolation, we have identified the formed compound structure.

引用

页码：200 / 204

页数：5

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