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- [21] Identification of Tricyclic Agonists of Sphingosine-1-phosphate Receptor 1 (S1P1) Employing Ligand-Based Drug DesignJOURNAL OF MEDICINAL CHEMISTRY, 2016, 59 (21) : 9837 - 9854Xiao, Hai-Yun论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Co, Res & Dev, POB 4000, Princeton, NJ 08543 USA Bristol Myers Squibb Co, Res & Dev, POB 4000, Princeton, NJ 08543 USAWatterson, Scott H.论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Co, Res & Dev, POB 4000, Princeton, NJ 08543 USA Bristol Myers Squibb Co, Res & Dev, POB 4000, Princeton, NJ 08543 USALangevine, Charles M.论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Co, Res & Dev, POB 4000, Princeton, NJ 08543 USA Bristol Myers Squibb Co, Res & Dev, POB 4000, Princeton, NJ 08543 USASrivastava, Anurag S.论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Co, Res & Dev, POB 4000, Princeton, NJ 08543 USA Bristol Myers Squibb Co, Res & Dev, POB 4000, Princeton, NJ 08543 USAKo, Soo S.论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Co, Res & Dev, POB 4000, Princeton, NJ 08543 USA Bristol Myers Squibb Co, Res & Dev, POB 4000, Princeton, NJ 08543 USAZhang, Yanlei论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Co, Res & Dev, POB 4000, Princeton, NJ 08543 USA Bristol Myers Squibb Co, Res & Dev, POB 4000, Princeton, NJ 08543 USACherney, Robert J.论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Co, Res & Dev, POB 4000, Princeton, NJ 08543 USA Bristol Myers Squibb Co, Res & Dev, POB 4000, Princeton, NJ 08543 USAGuo, Wei-Wei论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Co, Res & Dev, POB 4000, Princeton, NJ 08543 USA Bristol Myers Squibb Co, Res & Dev, POB 4000, Princeton, NJ 08543 USAGilmore, John L.论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Co, Res & Dev, POB 4000, Princeton, NJ 08543 USA Bristol Myers Squibb Co, Res & Dev, POB 4000, Princeton, NJ 08543 USAII, James E. Sheppeck论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Co, Res & Dev, POB 4000, Princeton, NJ 08543 USA Bristol Myers Squibb Co, Res & Dev, POB 4000, Princeton, NJ 08543 USAWu, Dauh-Rurng论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Co, Res & Dev, POB 4000, Princeton, NJ 08543 USA Bristol Myers Squibb Co, Res & Dev, POB 4000, Princeton, NJ 08543 USALi, Peng论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Co, Res & Dev, POB 4000, Princeton, NJ 08543 USA Bristol Myers Squibb Co, Res & Dev, POB 4000, Princeton, NJ 08543 USARamasamy, Duraisamy论文数: 0 引用数: 0 h-index: 0机构: BMS Biocon Res Ctr, Bangalore 560099, Karnataka, India Bristol Myers Squibb Co, Res & Dev, POB 4000, Princeton, NJ 08543 USAArunachalam, Piramanayagam论文数: 0 引用数: 0 h-index: 0机构: BMS Biocon Res Ctr, Bangalore 560099, Karnataka, India Bristol Myers Squibb Co, Res & Dev, POB 4000, Princeton, NJ 08543 USAMathur, Arvind论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Co, Res & Dev, POB 4000, Princeton, NJ 08543 USA Bristol Myers Squibb Co, Res & Dev, POB 4000, Princeton, NJ 08543 USATaylor, Tracy L.论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Co, Res & Dev, POB 4000, Princeton, NJ 08543 USA Bristol Myers Squibb Co, Res & Dev, POB 4000, Princeton, NJ 08543 USAShuster, David J.论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Co, Res & Dev, POB 4000, Princeton, NJ 08543 USA Bristol Myers Squibb Co, Res & Dev, POB 4000, Princeton, NJ 08543 USAMcIntyre, Kim W.论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Co, Res & Dev, POB 4000, Princeton, NJ 08543 USA Bristol Myers Squibb Co, Res & Dev, POB 4000, Princeton, NJ 08543 USAShen, Ding-Ren论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Co, Res & Dev, POB 4000, Princeton, NJ 08543 USA Bristol Myers Squibb Co, Res & Dev, POB 4000, Princeton, NJ 08543 USAYarde, Melissa论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Co, Res & Dev, POB 4000, Princeton, NJ 08543 USA Bristol Myers Squibb Co, Res & Dev, POB 4000, Princeton, NJ 08543 USACvijic, Mary Ellen论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Co, Res & Dev, POB 4000, Princeton, NJ 08543 USA Bristol Myers Squibb Co, Res & Dev, POB 4000, Princeton, NJ 08543 USAMarino, Anthony M.论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Co, Res & Dev, POB 4000, Princeton, NJ 08543 USA Bristol Myers Squibb Co, Res & Dev, POB 4000, Princeton, NJ 08543 USABalimane, Praveen V.论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Co, Res & Dev, POB 4000, Princeton, NJ 08543 USA Bristol Myers Squibb Co, Res & Dev, POB 4000, Princeton, NJ 08543 USAYang, Zheng论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Co, Res & Dev, POB 4000, Princeton, NJ 08543 USA Bristol Myers Squibb Co, Res & Dev, POB 4000, Princeton, NJ 08543 USABanas, Dana M.论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Co, Res & Dev, POB 4000, Princeton, NJ 08543 USA Bristol Myers Squibb Co, Res & Dev, POB 4000, Princeton, NJ 08543 USACornelius, Georgia论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Co, Res & Dev, POB 4000, Princeton, NJ 08543 USA Bristol Myers Squibb Co, Res & Dev, POB 4000, Princeton, NJ 08543 USAD'Arienzo, Celia J.论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Co, Res & Dev, POB 4000, Princeton, NJ 08543 USA Bristol Myers Squibb Co, Res & Dev, POB 4000, Princeton, NJ 08543 USAWarrack, Bethanne M.论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Co, Res & Dev, POB 4000, Princeton, NJ 08543 USA Bristol Myers Squibb Co, Res & Dev, POB 4000, Princeton, NJ 08543 USALehman-McKeeman, Lois论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Co, Res & Dev, POB 4000, Princeton, NJ 08543 USA Bristol Myers Squibb Co, Res & Dev, POB 4000, Princeton, NJ 08543 USASalter-Cid, Luisa M.论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Co, Res & Dev, POB 4000, Princeton, NJ 08543 USA Bristol Myers Squibb Co, Res & Dev, POB 4000, Princeton, NJ 08543 USAXie, Jenny论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Co, Res & Dev, POB 4000, Princeton, NJ 08543 USA Bristol Myers Squibb Co, Res & Dev, POB 4000, Princeton, NJ 08543 USABarrish, Joel C.论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Co, Res & Dev, POB 4000, Princeton, NJ 08543 USA Bristol Myers Squibb Co, Res & Dev, POB 4000, Princeton, NJ 08543 USACarter, Percy H.论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Co, Res & Dev, POB 4000, Princeton, NJ 08543 USA Bristol Myers Squibb Co, Res & Dev, POB 4000, Princeton, NJ 08543 USADyckman, Alaric J.论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Co, Res & Dev, POB 4000, Princeton, NJ 08543 USA Bristol Myers Squibb Co, Res & Dev, POB 4000, Princeton, NJ 08543 USADhar, T. G. Murali论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Co, Res & Dev, POB 4000, Princeton, NJ 08543 USA Bristol Myers Squibb Co, Res & Dev, POB 4000, Princeton, NJ 08543 USA
- [22] Discovery of Novel 1,2,4-Thiadiazole Derivatives as Potent, Orally Active Agonists of Sphingosine 1-Phosphate Receptor Subtype 1 (S1P1)JOURNAL OF MEDICINAL CHEMISTRY, 2012, 55 (09) : 4286 - 4296Ren, Feng论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline, R&D China, Shanghai 201203, Peoples R China GlaxoSmithKline, R&D China, Shanghai 201203, Peoples R ChinaDeng, Guanghui论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline, R&D China, Shanghai 201203, Peoples R China GlaxoSmithKline, R&D China, Shanghai 201203, Peoples R ChinaWang, Hailong论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline, R&D China, Shanghai 201203, Peoples R China GlaxoSmithKline, R&D China, Shanghai 201203, Peoples R ChinaLuan, Linbo论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline, R&D China, Shanghai 201203, Peoples R China GlaxoSmithKline, R&D China, Shanghai 201203, Peoples R ChinaMeng, Qinghua论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline, R&D China, Shanghai 201203, Peoples R China GlaxoSmithKline, R&D China, Shanghai 201203, Peoples R ChinaXu, Qiongfeng论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline, R&D China, Shanghai 201203, Peoples R China GlaxoSmithKline, R&D China, Shanghai 201203, Peoples R ChinaXu, Heng论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline, R&D China, Shanghai 201203, Peoples R China GlaxoSmithKline, R&D China, Shanghai 201203, Peoples R ChinaXu, Xuesong论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline, R&D China, Shanghai 201203, Peoples R China GlaxoSmithKline, R&D China, Shanghai 201203, Peoples R ChinaZhang, Haibo论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline, R&D China, Shanghai 201203, Peoples R China GlaxoSmithKline, R&D China, Shanghai 201203, Peoples R ChinaZhao, Baowei论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline, R&D China, Shanghai 201203, Peoples R China GlaxoSmithKline, R&D China, Shanghai 201203, Peoples R ChinaLi, Chengyong论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline, R&D China, Shanghai 201203, Peoples R China GlaxoSmithKline, R&D China, Shanghai 201203, Peoples R ChinaGuo, Taylor B.论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline, R&D China, Shanghai 201203, Peoples R China GlaxoSmithKline, R&D China, Shanghai 201203, Peoples R ChinaYang, Jiansong论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline, R&D China, Shanghai 201203, Peoples R China GlaxoSmithKline, R&D China, Shanghai 201203, Peoples R ChinaZhang, Wei论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline, R&D China, Shanghai 201203, Peoples R China GlaxoSmithKline, R&D China, Shanghai 201203, Peoples R ChinaZhao, Yonggang论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline, R&D China, Shanghai 201203, Peoples R China GlaxoSmithKline, R&D China, Shanghai 201203, Peoples R ChinaJia, Qiantao论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline, R&D China, Shanghai 201203, Peoples R China GlaxoSmithKline, R&D China, Shanghai 201203, Peoples R ChinaLu, Hongtao论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline, R&D China, Shanghai 201203, Peoples R China GlaxoSmithKline, R&D China, Shanghai 201203, Peoples R ChinaXiang, Jia-Ning论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline, R&D China, Shanghai 201203, Peoples R China GlaxoSmithKline, R&D China, Shanghai 201203, Peoples R ChinaElliott, John D.论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline, R&D China, Shanghai 201203, Peoples R China GlaxoSmithKline, R&D China, Shanghai 201203, Peoples R ChinaLin, Xichen论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline, R&D China, Shanghai 201203, Peoples R China GlaxoSmithKline, R&D China, Shanghai 201203, Peoples R China
- [23] Discovery of a novel class of zwitterionic, potent, selective and orally active S1P1 direct agonistsBIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2012, 22 (24) : 7672 - 7676Aguilar, Nuria论文数: 0 引用数: 0 h-index: 0机构: Labs Almirall SA, Almirall Res Ctr, E-08980 Barcelona, Spain Labs Almirall SA, Almirall Res Ctr, E-08980 Barcelona, SpainMir, Marta论文数: 0 引用数: 0 h-index: 0机构: Labs Almirall SA, Almirall Res Ctr, E-08980 Barcelona, Spain Labs Almirall SA, Almirall Res Ctr, E-08980 Barcelona, SpainGrima, Pedro M.论文数: 0 引用数: 0 h-index: 0机构: R&D&I Ctr, Ferrer Grp, E-08028 Barcelona, Spain Labs Almirall SA, Almirall Res Ctr, E-08980 Barcelona, SpainLopez, Manel论文数: 0 引用数: 0 h-index: 0机构: Labs Almirall SA, Almirall Res Ctr, E-08980 Barcelona, Spain Labs Almirall SA, Almirall Res Ctr, E-08980 Barcelona, SpainSegarra, Victor论文数: 0 引用数: 0 h-index: 0机构: Labs Almirall SA, Almirall Res Ctr, E-08980 Barcelona, Spain Labs Almirall SA, Almirall Res Ctr, E-08980 Barcelona, SpainEsteban, Laia论文数: 0 引用数: 0 h-index: 0机构: Dukechem, E-08799 Barcelona, Spain Labs Almirall SA, Almirall Res Ctr, E-08980 Barcelona, SpainMoreno, Imma论文数: 0 引用数: 0 h-index: 0机构: Labs Almirall SA, Almirall Res Ctr, E-08980 Barcelona, Spain Labs Almirall SA, Almirall Res Ctr, E-08980 Barcelona, SpainGodessart, Nuria论文数: 0 引用数: 0 h-index: 0机构: Labs Almirall SA, Almirall Res Ctr, E-08980 Barcelona, Spain Labs Almirall SA, Almirall Res Ctr, E-08980 Barcelona, SpainTarrason, Gema论文数: 0 引用数: 0 h-index: 0机构: Labs Almirall SA, Almirall Res Ctr, E-08980 Barcelona, Spain Labs Almirall SA, Almirall Res Ctr, E-08980 Barcelona, SpainDomenech, Teresa论文数: 0 引用数: 0 h-index: 0机构: Labs Almirall SA, Almirall Res Ctr, E-08980 Barcelona, Spain Labs Almirall SA, Almirall Res Ctr, E-08980 Barcelona, SpainVilella, Dolors论文数: 0 引用数: 0 h-index: 0机构: Labs Almirall SA, Almirall Res Ctr, E-08980 Barcelona, Spain Labs Almirall SA, Almirall Res Ctr, E-08980 Barcelona, SpainArmengol, Clara论文数: 0 引用数: 0 h-index: 0机构: Labs Almirall SA, Almirall Res Ctr, E-08980 Barcelona, Spain Labs Almirall SA, Almirall Res Ctr, E-08980 Barcelona, SpainCordoba, Monica论文数: 0 引用数: 0 h-index: 0机构: Labs Almirall SA, Almirall Res Ctr, E-08980 Barcelona, Spain Labs Almirall SA, Almirall Res Ctr, E-08980 Barcelona, SpainSabate, Mar论文数: 0 引用数: 0 h-index: 0机构: Labs Almirall SA, Almirall Res Ctr, E-08980 Barcelona, Spain Labs Almirall SA, Almirall Res Ctr, E-08980 Barcelona, SpainCasals, Daniel论文数: 0 引用数: 0 h-index: 0机构: Labs Almirall SA, Almirall Res Ctr, E-08980 Barcelona, Spain Labs Almirall SA, Almirall Res Ctr, E-08980 Barcelona, SpainDominguez, Maria论文数: 0 引用数: 0 h-index: 0机构: Labs Almirall SA, Almirall Res Ctr, E-08980 Barcelona, Spain Labs Almirall SA, Almirall Res Ctr, E-08980 Barcelona, Spain
- [24] Indole-propionic acid derivatives as potent, S1P3-sparing and EAE efficacious sphingosine-1-phosphate 1 (S1P1) receptor agonistsBIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2012, 22 (08) : 2794 - 2797Meng, Qinghua论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline, Res & Dev, Shanghai 201023, Peoples R China GlaxoSmithKline, Res & Dev, Shanghai 201023, Peoples R ChinaZhao, Baowei论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline, Res & Dev, Shanghai 201023, Peoples R China GlaxoSmithKline, Res & Dev, Shanghai 201023, Peoples R ChinaXu, Qiongfeng论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline, Res & Dev, Shanghai 201023, Peoples R China GlaxoSmithKline, Res & Dev, Shanghai 201023, Peoples R ChinaXu, Xuesong论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline, Res & Dev, Shanghai 201023, Peoples R China GlaxoSmithKline, Res & Dev, Shanghai 201023, Peoples R ChinaDeng, Guanghui论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline, Res & Dev, Shanghai 201023, Peoples R China GlaxoSmithKline, Res & Dev, Shanghai 201023, Peoples R ChinaLi, Chengyong论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline, Res & Dev, Shanghai 201023, Peoples R China GlaxoSmithKline, Res & Dev, Shanghai 201023, Peoples R ChinaLuan, Linbo论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline, Res & Dev, Shanghai 201023, Peoples R China GlaxoSmithKline, Res & Dev, Shanghai 201023, Peoples R ChinaRen, Feng论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline, Res & Dev, Shanghai 201023, Peoples R China GlaxoSmithKline, Res & Dev, Shanghai 201023, Peoples R ChinaWang, Hailong论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline, Res & Dev, Shanghai 201023, Peoples R China GlaxoSmithKline, Res & Dev, Shanghai 201023, Peoples R ChinaXu, Heng论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline, Res & Dev, Shanghai 201023, Peoples R China GlaxoSmithKline, Res & Dev, Shanghai 201023, Peoples R ChinaXu, Yan论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline, Res & Dev, Shanghai 201023, Peoples R China GlaxoSmithKline, Res & Dev, Shanghai 201023, Peoples R ChinaZhang, Haibo论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline, Res & Dev, Shanghai 201023, Peoples R China GlaxoSmithKline, Res & Dev, Shanghai 201023, Peoples R ChinaXiang, Jia-Ning论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline, Res & Dev, Shanghai 201023, Peoples R China GlaxoSmithKline, Res & Dev, Shanghai 201023, Peoples R ChinaElliott, John D.论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline, Res & Dev, Shanghai 201023, Peoples R China GlaxoSmithKline, Res & Dev, Shanghai 201023, Peoples R ChinaGuo, Taylor B.论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline, Res & Dev, Shanghai 201023, Peoples R China GlaxoSmithKline, Res & Dev, Shanghai 201023, Peoples R ChinaZhao, Yonggang论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline, Res & Dev, Shanghai 201023, Peoples R China GlaxoSmithKline, Res & Dev, Shanghai 201023, Peoples R ChinaZhang, Wei论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline, Res & Dev, Shanghai 201023, Peoples R China GlaxoSmithKline, Res & Dev, Shanghai 201023, Peoples R ChinaLu, Hongtao论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline, Res & Dev, Shanghai 201023, Peoples R China GlaxoSmithKline, Res & Dev, Shanghai 201023, Peoples R ChinaLin, Xichen论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline, Res & Dev, Shanghai 201023, Peoples R China GlaxoSmithKline, Res & Dev, Shanghai 201023, Peoples R China
- [25] Discovery of AMG 369, a potent and selective thiazolo[5,4-b]pyridine agonist of sphingosine-1-phosphate receptors 1 and 5 (S1P1 and S1P5)ABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY, 2011, 241Gee, Victor J.论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Dept Med Chem, Thousand Oaks, CA USA Amgen Inc, Dept Med Chem, Thousand Oaks, CA USA
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