Synthesis of some new 2-substituted-4-sulfamoylphenylazo-thiophene and/or thiazole derivatives as antibacterial agents

被引：11

作者：

Fadda, Ahmed A. ^{[1
]}

El-badraw, Afnan M. ^{[1
]}

Refat, Hala M. ^{[2
]}

Abdel-Latif, Ehab ^{[1
]}

机构：

[1] Mansoura Univ, Fac Sci, Dept Chem, ET-35516 Mansoura, Egypt

[2] Suez Canal Univ, Fac Sci, Dept Chem, Al Arish, Egypt

来源：

PHOSPHORUS SULFUR AND SILICON AND THE RELATED ELEMENTS | 2016年 / 191卷 / 05期

关键词：

Benzoylacetone; sulfanilamide; thiocarbamoyl; thiophene; thiazolodin-5-one; antibacterial activities; DESIGN;

D O I：

10.1080/10426507.2015.1100183

中图分类号：

O61 [无机化学];

学科分类号：

070301 ; 081704 ;

摘要：

Benzaylacetone has been reacted with phenyl Isothaacyanate to afford two difFerent thiocarbarnoyl derive tines (alpha-phenylthiocarbamoyl benzoy acetone arid benzo3d thioacetanilide) depending upon the bas used to perforrri the reaction. Several new 2-substituted-4-sulfamoylpheriylazo-thiapherie and/or thiazole derivatives were synthesized by heterocyclization of the thiocarbarnoyl derivatives with various halogenated reagents. The synthesized compounds were screened fortheir antibacterial activities; they showed accepted activities with respect to the control drugs.

引用

页码：778 / 785

页数：8

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