SYNTHESIS AND BIOLOGICAL ACTIVITY OF N-{5-(4-METHYLPHENYL) DIAZENYL-4-PHENYL-1, 3-THIAZOL-2-YL}BENZAMIDE DERIVATIVES

被引：0

作者：

Prajapati, Ashishkumar Kantilal ^{[1
]}

Modi, Vishal Pankajkumar ^{[1
]}

机构：

[1] Maharaja Sayajirao Univ Baroda, Fac Engn & Technol, Dept Appl Chem, Vadodara 390001, Gujarat, India

来源：

QUIMICA NOVA | 2011年 / 34卷 / 05期

关键词：

aminothiazole derivatives; amide linkage; microbial activity; ANTIMICROBIAL ACTIVITY; POTENTIAL ANTINEOPLASTICS; THIAZOLE; AGENTS; DESIGN; QSAR;

D O I：

暂无

中图分类号：

O6 [化学];

学科分类号：

0703 ;

摘要：

In the present study, various amides of 2-amino-5-(4-methylphenyl)-diazenyl-4-phenyl-1, 3-thiazole was synthesized and their biological activities were evaluated. All the synthesized compounds were characterized by the combination of elemental analysis and standard spectroscopic methods. They are screened for anti-bacterial activity against Escherichia coli and Staphylococcus aureus as well as screened for antifungal activity against Aspergillus niger and Apergillus oryzae by cup plate method at 1 mu g/mL concentration in DMF.

引用

页码：771 / 774

页数：4

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