A NEW ENTRY FOR PREPARATION OF 2-SUBSTITUTED AZAINDOLES

被引：6
|
作者：
Shaykoon, Montaser [1 ]
Shaykoon, Ahmed [1 ]
Inagaki, Fuyuhiko [1 ]
Mukai, Chisato [1 ]
机构：
[1] Kanazawa Univ, Grad Sch Nat Sci & Technol, Div Pharmaceut Sci, Kanazawa, Ishikawa 9201192, Japan
来源：
HETEROCYCLES | 2010年 / 80卷 / 01期
关键词：
2-Substituted; 5-; 6-and; 7-Azaindoles; 3-Substituted Allenylstannane; Iodoaminopyridine; Stille Coupling; Cyclization; MAP KINASE; RWJ; 68354; 6-AZAINDOLES; P38; 5-AZAINDOLES; 4-AZAINDOLES; DERIVATIVES; REACTIVITY; INHIBITOR; REAGENTS;
D O I：
10.3987/COM-09-S(S)29
中图分类号：
O62 [有机化学];
学科分类号：
070303 ; 081704 ;
摘要：
A series of 2-substituted 5-, 6- and 7-azaindoles were synthesized from iodo-N-(tert-butoxycarbonyl)aminopyridines via the corresponding allenyl derivatives.
引用
收藏
页码：133 / 139
页数：7
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