Synthesis of C-14-Labeled levamisole and C-13-labeled tetramisole

被引：0

作者：

Feil, VJ

机构：

来源：

JOURNAL OF LABELLED COMPOUNDS & RADIOPHARMACEUTICALS | 1996年 / 38卷 / 12期

关键词：

C-14]levamisole; C-13]tetramisole; -]-2,3,5,6-tetrahydro-6-phenyl[C-14-UL]imidazo[2,1-b]thiazole [+/-]-2,3,5,6-tetrahydro-6-phenyl[C-13(6)]imidazo[2,1-b]-thiazole;

D O I：

暂无

中图分类号：

Q5 [生物化学];

学科分类号：

071010 ; 081704 ;

摘要：

The syntheses of C-14-ring labeled levamisole ([-]-2,3,5,6-tetrahydro-6-phenyl[C-14-UL]imidazo[2,1-b] thiazole) from acetophenone-ring-UL-C-14 in 5 steps plus resolution with a 7.5% overall yield, and C-13(6)-ring labeled tetramisole ([+/-]-2,3,5,6-tetrahydro-6-phenyl[C-13(6)]imidazo[2,1-b] thiazole) from benzene-C-13(6) in 6 steps with a 9.0% overall yield are described.

引用

页码：1071 / 1076

页数：6

共 7 条

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