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- [1] Design, synthesis, and structure-activity relationship of novel CCR2 antagonistsBIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2009, 19 (06) : 1830 - 1834Kothandaraman, Shankaran论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Dept Med Chem, Rahway, NJ 07065 USA Merck Res Labs, Dept Med Chem, Rahway, NJ 07065 USADonnely, Karla L.论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Dept Med Chem, Rahway, NJ 07065 USA Merck Res Labs, Dept Med Chem, Rahway, NJ 07065 USAButora, Gabor论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Dept Med Chem, Rahway, NJ 07065 USA Merck Res Labs, Dept Med Chem, Rahway, NJ 07065 USAJiao, Richard论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Dept Med Chem, Rahway, NJ 07065 USA Merck Res Labs, Dept Med Chem, Rahway, NJ 07065 USAPasternak, Alexander论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Dept Med Chem, Rahway, NJ 07065 USA Merck Res Labs, Dept Med Chem, Rahway, NJ 07065 USAMorriello, Gregori J.论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Dept Med Chem, Rahway, NJ 07065 USA Merck Res Labs, Dept Med Chem, Rahway, NJ 07065 USAGoble, Stephen D.论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Dept Med Chem, Rahway, NJ 07065 USA Merck Res Labs, Dept Med Chem, Rahway, NJ 07065 USAZhou, Changyou论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Dept Med Chem, Rahway, NJ 07065 USA Merck Res Labs, Dept Med Chem, Rahway, NJ 07065 USAMills, Sander G.论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Dept Med Chem, Rahway, NJ 07065 USA Merck Res Labs, Dept Med Chem, Rahway, NJ 07065 USAMacCoss, Malcolm论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Dept Med Chem, Rahway, NJ 07065 USA Merck Res Labs, Dept Med Chem, Rahway, NJ 07065 USAVicario, Pasquale P.论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Dept Immunol, Rahway, NJ 07065 USA Merck Res Labs, Dept Med Chem, Rahway, NJ 07065 USAAyala, Julia M.论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Dept Immunol, Rahway, NJ 07065 USA Merck Res Labs, Dept Med Chem, Rahway, NJ 07065 USADeMartino, Julie A.论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Dept Immunol, Rahway, NJ 07065 USA Merck Res Labs, Dept Med Chem, Rahway, NJ 07065 USAStruthers, Mary论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Dept Immunol, Rahway, NJ 07065 USA Merck Res Labs, Dept Med Chem, Rahway, NJ 07065 USACascieri, Margaret A.论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Dept Immunol, Rahway, NJ 07065 USA Merck Res Labs, Dept Med Chem, Rahway, NJ 07065 USAYang, Lihu论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Dept Med Chem, Rahway, NJ 07065 USA Merck Res Labs, Dept Med Chem, Rahway, NJ 07065 USA
- [2] Design and synthesis of novel small molecule CCR2 antagonists: Evaluation of 4-aminopiperidine derivativesBIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2014, 24 (23) : 5377 - 5380Vilums, M.论文数: 0 引用数: 0 h-index: 0机构: Leiden Univ, Leiden Acad Ctr Drug Res, Div Med Chem, NL-2300 RA Leiden, Netherlands Leiden Univ, Leiden Acad Ctr Drug Res, Div Med Chem, NL-2300 RA Leiden, NetherlandsZweemer, A. J. M.论文数: 0 引用数: 0 h-index: 0机构: Leiden Univ, Leiden Acad Ctr Drug Res, Div Med Chem, NL-2300 RA Leiden, Netherlands Leiden Univ, Leiden Acad Ctr Drug Res, Div Med Chem, NL-2300 RA Leiden, NetherlandsDekkers, S.论文数: 0 引用数: 0 h-index: 0机构: Leiden Univ, Leiden Acad Ctr Drug Res, Div Med Chem, NL-2300 RA Leiden, Netherlands Leiden Univ, Leiden Acad Ctr Drug Res, Div Med Chem, NL-2300 RA Leiden, NetherlandsAskar, Y.论文数: 0 引用数: 0 h-index: 0机构: Leiden Univ, Leiden Acad Ctr Drug Res, Div Med Chem, NL-2300 RA Leiden, Netherlands Leiden Univ, Leiden Acad Ctr Drug Res, Div Med Chem, NL-2300 RA Leiden, Netherlandsde Vries, H.论文数: 0 引用数: 0 h-index: 0机构: Leiden Univ, Leiden Acad Ctr Drug Res, Div Med Chem, NL-2300 RA Leiden, Netherlands Leiden Univ, Leiden Acad Ctr Drug Res, Div Med Chem, NL-2300 RA Leiden, NetherlandsSaunders, J.论文数: 0 引用数: 0 h-index: 0机构: Vertex Pharmaceut Inc, San Diego, CA USA Leiden Univ, Leiden Acad Ctr Drug Res, Div Med Chem, NL-2300 RA Leiden, NetherlandsStamos, D.论文数: 0 引用数: 0 h-index: 0机构: Vertex Pharmaceut Inc, San Diego, CA USA Leiden Univ, Leiden Acad Ctr Drug Res, Div Med Chem, NL-2300 RA Leiden, NetherlandsBrussee, J.论文数: 0 引用数: 0 h-index: 0机构: Leiden Univ, Leiden Acad Ctr Drug Res, Div Med Chem, NL-2300 RA Leiden, Netherlands Leiden Univ, Leiden Acad Ctr Drug Res, Div Med Chem, NL-2300 RA Leiden, NetherlandsHeitman, L. H.论文数: 0 引用数: 0 h-index: 0机构: Leiden Univ, Leiden Acad Ctr Drug Res, Div Med Chem, NL-2300 RA Leiden, Netherlands Leiden Univ, Leiden Acad Ctr Drug Res, Div Med Chem, NL-2300 RA Leiden, NetherlandsIJzerman, A. P.论文数: 0 引用数: 0 h-index: 0机构: Leiden Univ, Leiden Acad Ctr Drug Res, Div Med Chem, NL-2300 RA Leiden, Netherlands Leiden Univ, Leiden Acad Ctr Drug Res, Div Med Chem, NL-2300 RA Leiden, Netherlands
- [3] α-Aminothiazole-γ-aminobutanoic amides as potent, small molecule CCR2 receptor antagonistsBIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2007, 17 (02) : 309 - 314Zhou, Changyou论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Dept Med Chem, Rahway, NJ 07065 USA Merck Res Labs, Dept Med Chem, Rahway, NJ 07065 USAGuo, Liangqin论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Dept Med Chem, Rahway, NJ 07065 USAParsons, William H.论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Dept Med Chem, Rahway, NJ 07065 USAMills, Sander G.论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Dept Med Chem, Rahway, NJ 07065 USAMacCoss, Malcolm论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Dept Med Chem, Rahway, NJ 07065 USAVicario, Pasquale P.论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Dept Med Chem, Rahway, NJ 07065 USAZweerink, Hans论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Dept Med Chem, Rahway, NJ 07065 USACascieri, Margaret A.论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Dept Med Chem, Rahway, NJ 07065 USASpringer, Martin S.论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Dept Med Chem, Rahway, NJ 07065 USAYang, Lihu论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Dept Med Chem, Rahway, NJ 07065 USA
- [4] MEDI 72-Design, synthesis and structure-activity relationship of novel CCR2 antagonistsABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY, 2008, 236Kothandaraman, Shankaran论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Dept Med Chem, Rahway, NJ 07065 USA Merck Res Labs, Dept Med Chem, Rahway, NJ 07065 USADonnely, Karla L.论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Dept Med Chem, Rahway, NJ 07065 USA Merck Res Labs, Dept Med Chem, Rahway, NJ 07065 USAJiao, Richard X.论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Dept Med Chem, Rahway, NJ 07065 USA Merck Res Labs, Dept Med Chem, Rahway, NJ 07065 USAButora, Gabor论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Dept Med Chem, Rahway, NJ 07065 USA Merck Res Labs, Dept Med Chem, Rahway, NJ 07065 USAPasternak, Alexander论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Dept Med Chem, Rahway, NJ 07065 USA Merck Res Labs, Dept Med Chem, Rahway, NJ 07065 USAMorriello, Gregori J.论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Dept Med Chem, Rahway, NJ 07065 USA Merck Res Labs, Dept Med Chem, Rahway, NJ 07065 USAGoble, Steve论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Dept Med Chem, Rahway, NJ 07065 USA Merck Res Labs, Dept Med Chem, Rahway, NJ 07065 USAZhou, Changyou论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Dept Med Chem, Rahway, NJ 07065 USA Merck Res Labs, Dept Med Chem, Rahway, NJ 07065 USAYang, Lihu论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Dept Med Chem, Rahway, NJ 07065 USA Merck Res Labs, Dept Med Chem, Rahway, NJ 07065 USAMills, Sander G.论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Dept Med Chem, Rahway, NJ 07065 USA Merck Res Labs, Dept Med Chem, Rahway, NJ 07065 USAMacCoss, Malcolm论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Dept Med Chem, Rahway, NJ 07065 USA Merck Res Labs, Dept Med Chem, Rahway, NJ 07065 USAAyala, Julia M.论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Dept Immunol, Rahway, NJ 07065 USA Merck Res Labs, Dept Med Chem, Rahway, NJ 07065 USAVicario, Pasquale P.论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Dept Immunol, Rahway, NJ 07065 USA Merck Res Labs, Dept Med Chem, Rahway, NJ 07065 USACascieri, Margaret A.论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Dept Immunol, Rahway, NJ 07065 USA Merck Res Labs, Dept Med Chem, Rahway, NJ 07065 USA
- [5] Pharmacophore Model-based Design and Synthesis of New Structure Small Molecule CCR2 InhibitorsACTA CHIMICA SINICA, 2015, 73 (07) : 679 - 684Qin Lihuai论文数: 0 引用数: 0 h-index: 0机构: Chinese Acad Sci, Shanghai Inst Mat Med, CAS Key Lab Receptor Res, Shanghai 201203, Peoples R China Chinese Acad Sci, Shanghai Inst Mat Med, CAS Key Lab Receptor Res, Shanghai 201203, Peoples R ChinaLi Xiaoguang论文数: 0 引用数: 0 h-index: 0机构: Chinese Acad Sci, Shanghai Inst Nutr Sci, CAS Key Lab Food Safety, Shanghai 200031, Peoples R China Chinese Acad Sci, Shanghai Inst Mat Med, CAS Key Lab Receptor Res, Shanghai 201203, Peoples R ChinaWang Zhilong论文数: 0 引用数: 0 h-index: 0机构: Chinese Acad Sci, Shanghai Inst Mat Med, CAS Key Lab Receptor Res, Shanghai 201203, Peoples R China Chinese Acad Sci, Shanghai Inst Mat Med, CAS Key Lab Receptor Res, Shanghai 201203, Peoples R ChinaYao Wenbo论文数: 0 引用数: 0 h-index: 0机构: Chinese Acad Sci, Shanghai Inst Nutr Sci, CAS Key Lab Food Safety, Shanghai 200031, Peoples R China Chinese Acad Sci, Shanghai Inst Mat Med, CAS Key Lab Receptor Res, Shanghai 201203, Peoples R ChinaWang Hui论文数: 0 引用数: 0 h-index: 0机构: Chinese Acad Sci, Shanghai Inst Nutr Sci, CAS Key Lab Food Safety, Shanghai 200031, Peoples R China Chinese Acad Sci, Shanghai Inst Mat Med, CAS Key Lab Receptor Res, Shanghai 201203, Peoples R ChinaXie Xin论文数: 0 引用数: 0 h-index: 0机构: Chinese Acad Sci, Shanghai Inst Mat Med, CAS Key Lab Receptor Res, Shanghai 201203, Peoples R China Chinese Acad Sci, Shanghai Inst Mat Med, CAS Key Lab Receptor Res, Shanghai 201203, Peoples R ChinaLong Yaqiu论文数: 0 引用数: 0 h-index: 0机构: Chinese Acad Sci, Shanghai Inst Mat Med, CAS Key Lab Receptor Res, Shanghai 201203, Peoples R China Chinese Acad Sci, Shanghai Inst Mat Med, CAS Key Lab Receptor Res, Shanghai 201203, Peoples R China
- [6] Synthesis, structure - Activity relationship and in vivo antiinflammatory efficacy of substituted dipiperidines as CCR2 antagonistsJOURNAL OF MEDICINAL CHEMISTRY, 2007, 50 (23) : 5561 - 5563Xia, Mingde论文数: 0 引用数: 0 h-index: 0机构: Johnson & Johnson Pharmaceut Res & Dev LLC, Drug Discovery, Cranbury, NJ 08512 USA Johnson & Johnson Pharmaceut Res & Dev LLC, Drug Discovery, Cranbury, NJ 08512 USAHou, Cuifen论文数: 0 引用数: 0 h-index: 0机构: Johnson & Johnson Pharmaceut Res & Dev LLC, Drug Discovery, Cranbury, NJ 08512 USA Johnson & Johnson Pharmaceut Res & Dev LLC, Drug Discovery, Cranbury, NJ 08512 USADeMong, Duane E.论文数: 0 引用数: 0 h-index: 0机构: Johnson & Johnson Pharmaceut Res & Dev LLC, Drug Discovery, Cranbury, NJ 08512 USA Johnson & Johnson Pharmaceut Res & Dev LLC, Drug Discovery, Cranbury, NJ 08512 USAPollack, Scott R.论文数: 0 引用数: 0 h-index: 0机构: Johnson & Johnson Pharmaceut Res & Dev LLC, Drug Discovery, Cranbury, NJ 08512 USA Johnson & Johnson Pharmaceut Res & Dev LLC, Drug Discovery, Cranbury, NJ 08512 USAPan, Meng论文数: 0 引用数: 0 h-index: 0机构: Johnson & Johnson Pharmaceut Res & Dev LLC, Drug Discovery, Cranbury, NJ 08512 USA Johnson & Johnson Pharmaceut Res & Dev LLC, Drug Discovery, Cranbury, NJ 08512 USABrackley, James A.论文数: 0 引用数: 0 h-index: 0机构: Johnson & Johnson Pharmaceut Res & Dev LLC, Drug Discovery, Cranbury, NJ 08512 USA Johnson & Johnson Pharmaceut Res & Dev LLC, Drug Discovery, Cranbury, NJ 08512 USAJain, Nareshkumar论文数: 0 引用数: 0 h-index: 0机构: Johnson & Johnson Pharmaceut Res & Dev LLC, Drug Discovery, Cranbury, NJ 08512 USA Johnson & Johnson Pharmaceut Res & Dev LLC, Drug Discovery, Cranbury, NJ 08512 USAGerchak, Chrissy论文数: 0 引用数: 0 h-index: 0机构: Johnson & Johnson Pharmaceut Res & Dev LLC, Drug Discovery, Cranbury, NJ 08512 USA Johnson & Johnson Pharmaceut Res & Dev LLC, Drug Discovery, Cranbury, NJ 08512 USASinger, Monica论文数: 0 引用数: 0 h-index: 0机构: Johnson & Johnson Pharmaceut Res & Dev LLC, Drug Discovery, Cranbury, NJ 08512 USA Johnson & Johnson Pharmaceut Res & Dev LLC, Drug Discovery, Cranbury, NJ 08512 USAMalaviya, Ravi论文数: 0 引用数: 0 h-index: 0机构: Johnson & Johnson Pharmaceut Res & Dev LLC, Drug Discovery, Cranbury, NJ 08512 USA Johnson & Johnson Pharmaceut Res & Dev LLC, Drug Discovery, Cranbury, NJ 08512 USAMatheis, Michele论文数: 0 引用数: 0 h-index: 0机构: Johnson & Johnson Pharmaceut Res & Dev LLC, Drug Discovery, Cranbury, NJ 08512 USA Johnson & Johnson Pharmaceut Res & Dev LLC, Drug Discovery, Cranbury, NJ 08512 USAOlini, Gil论文数: 0 引用数: 0 h-index: 0机构: Johnson & Johnson Pharmaceut Res & Dev LLC, Drug Discovery, Cranbury, NJ 08512 USA Johnson & Johnson Pharmaceut Res & Dev LLC, Drug Discovery, Cranbury, NJ 08512 USACavender, Druie论文数: 0 引用数: 0 h-index: 0机构: Johnson & Johnson Pharmaceut Res & Dev LLC, Drug Discovery, Cranbury, NJ 08512 USA Johnson & Johnson Pharmaceut Res & Dev LLC, Drug Discovery, Cranbury, NJ 08512 USAWachter, Michael论文数: 0 引用数: 0 h-index: 0机构: Johnson & Johnson Pharmaceut Res & Dev LLC, Drug Discovery, Cranbury, NJ 08512 USA Johnson & Johnson Pharmaceut Res & Dev LLC, Drug Discovery, Cranbury, NJ 08512 USA
- [7] Synthesis and structure-activity relationship of 7-azaindole piperidine derivatives as CCR2 antagonistsBIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2008, 18 (24) : 6468 - 6470Xia, Mingde论文数: 0 引用数: 0 h-index: 0机构: Johnson & Johnson Pharmaceut Res & Dev LLC, Drug Discovery, Cranbury, NJ 08512 USA Johnson & Johnson Pharmaceut Res & Dev LLC, Drug Discovery, Cranbury, NJ 08512 USAHou, Cuifen论文数: 0 引用数: 0 h-index: 0机构: Johnson & Johnson Pharmaceut Res & Dev LLC, Drug Discovery, Cranbury, NJ 08512 USA Johnson & Johnson Pharmaceut Res & Dev LLC, Drug Discovery, Cranbury, NJ 08512 USADeMong, Duane论文数: 0 引用数: 0 h-index: 0机构: Johnson & Johnson Pharmaceut Res & Dev LLC, Drug Discovery, Cranbury, NJ 08512 USA Johnson & Johnson Pharmaceut Res & Dev LLC, Drug Discovery, Cranbury, NJ 08512 USAPollack, Scott论文数: 0 引用数: 0 h-index: 0机构: Johnson & Johnson Pharmaceut Res & Dev LLC, Drug Discovery, Cranbury, NJ 08512 USA Johnson & Johnson Pharmaceut Res & Dev LLC, Drug Discovery, Cranbury, NJ 08512 USAPan, Meng论文数: 0 引用数: 0 h-index: 0机构: Johnson & Johnson Pharmaceut Res & Dev LLC, Drug Discovery, Cranbury, NJ 08512 USA Johnson & Johnson Pharmaceut Res & Dev LLC, Drug Discovery, Cranbury, NJ 08512 USASinger, Monica论文数: 0 引用数: 0 h-index: 0机构: Johnson & Johnson Pharmaceut Res & Dev LLC, Drug Discovery, Cranbury, NJ 08512 USA Johnson & Johnson Pharmaceut Res & Dev LLC, Drug Discovery, Cranbury, NJ 08512 USAMatheis, Michele论文数: 0 引用数: 0 h-index: 0机构: Johnson & Johnson Pharmaceut Res & Dev LLC, Drug Discovery, Cranbury, NJ 08512 USA Johnson & Johnson Pharmaceut Res & Dev LLC, Drug Discovery, Cranbury, NJ 08512 USAMurray, William论文数: 0 引用数: 0 h-index: 0机构: Johnson & Johnson Pharmaceut Res & Dev LLC, Drug Discovery, Cranbury, NJ 08512 USA Johnson & Johnson Pharmaceut Res & Dev LLC, Drug Discovery, Cranbury, NJ 08512 USACavender, Druie论文数: 0 引用数: 0 h-index: 0机构: Johnson & Johnson Pharmaceut Res & Dev LLC, Drug Discovery, Cranbury, NJ 08512 USA Johnson & Johnson Pharmaceut Res & Dev LLC, Drug Discovery, Cranbury, NJ 08512 USAWachter, Michael论文数: 0 引用数: 0 h-index: 0机构: Johnson & Johnson Pharmaceut Res & Dev LLC, Drug Discovery, Cranbury, NJ 08512 USA Johnson & Johnson Pharmaceut Res & Dev LLC, Drug Discovery, Cranbury, NJ 08512 USA
- [8] Structure-Affinity and Structure-Kinetic Relationship Studies of Benzodiazepine Derivatives for the Development of Efficacious Vasopressin V2 Receptor AntagonistsJOURNAL OF MEDICINAL CHEMISTRY, 2023, 66 (05) : 3621 - 3634Cao, Xudong论文数: 0 引用数: 0 h-index: 0机构: Xuzhou Med Univ, Jiangsu Key Lab New Drug Res & Clin Pharm, Xuzhou 221004, Jiangsu, Peoples R China Xuzhou Med Univ, Jiangsu Key Lab New Drug Res & Clin Pharm, Xuzhou 221004, Jiangsu, Peoples R ChinaWang, Peng论文数: 0 引用数: 0 h-index: 0机构: Xuzhou Med Univ, Jiangsu Key Lab New Drug Res & Clin Pharm, Xuzhou 221004, Jiangsu, Peoples R China Xuzhou Med Univ, Jiangsu Key Lab New Drug Res & Clin Pharm, Xuzhou 221004, Jiangsu, Peoples R ChinaZhao, Wenchao论文数: 0 引用数: 0 h-index: 0机构: Xuzhou Med Univ, Jiangsu Key Lab New Drug Res & Clin Pharm, Xuzhou 221004, Jiangsu, Peoples R China Xuzhou Med Univ, Jiangsu Key Lab New Drug Res & Clin Pharm, Xuzhou 221004, Jiangsu, Peoples R ChinaYuan, Haoxing论文数: 0 引用数: 0 h-index: 0机构: Xuzhou Med Univ, Jiangsu Key Lab New Drug Res & Clin Pharm, Xuzhou 221004, Jiangsu, Peoples R China Xuzhou Med Univ, Jiangsu Key Lab New Drug Res & Clin Pharm, Xuzhou 221004, Jiangsu, Peoples R ChinaHu, Hongtao论文数: 0 引用数: 0 h-index: 0机构: Xuzhou Med Univ, Jiangsu Key Lab New Drug Res & Clin Pharm, Xuzhou 221004, Jiangsu, Peoples R China Xuzhou Med Univ, Jiangsu Key Lab New Drug Res & Clin Pharm, Xuzhou 221004, Jiangsu, Peoples R ChinaChen, Ting论文数: 0 引用数: 0 h-index: 0机构: Xuzhou Med Univ, Jiangsu Key Lab New Drug Res & Clin Pharm, Xuzhou 221004, Jiangsu, Peoples R China Xuzhou Med Univ, Jiangsu Key Lab New Drug Res & Clin Pharm, Xuzhou 221004, Jiangsu, Peoples R ChinaZhang, Yixiao论文数: 0 引用数: 0 h-index: 0机构: Xuzhou Med Univ, Jiangsu Key Lab New Drug Res & Clin Pharm, Xuzhou 221004, Jiangsu, Peoples R China Xuzhou Med Univ, Jiangsu Key Lab New Drug Res & Clin Pharm, Xuzhou 221004, Jiangsu, Peoples R ChinaRen, Ying论文数: 0 引用数: 0 h-index: 0机构: Xuzhou Med Univ, Jiangsu Key Lab New Drug Res & Clin Pharm, Xuzhou 221004, Jiangsu, Peoples R China Xuzhou Med Univ, Jiangsu Key Lab New Drug Res & Clin Pharm, Xuzhou 221004, Jiangsu, Peoples R ChinaSu, Limin论文数: 0 引用数: 0 h-index: 0机构: Xuzhou Med Univ, Jiangsu Key Lab New Drug Res & Clin Pharm, Xuzhou 221004, Jiangsu, Peoples R China Xuzhou Med Univ, Jiangsu Key Lab New Drug Res & Clin Pharm, Xuzhou 221004, Jiangsu, Peoples R ChinaFu, Kequan论文数: 0 引用数: 0 h-index: 0机构: Xuzhou Med Univ, Jiangsu Key Lab New Drug Res & Clin Pharm, Xuzhou 221004, Jiangsu, Peoples R China Xuzhou Med Univ, Jiangsu Key Lab New Drug Res & Clin Pharm, Xuzhou 221004, Jiangsu, Peoples R ChinaLiu, Hongli论文数: 0 引用数: 0 h-index: 0机构: Xuzhou Med Univ, Jiangsu Key Lab New Drug Res & Clin Pharm, Xuzhou 221004, Jiangsu, Peoples R China Xuzhou Med Univ, Jiangsu Key Lab New Drug Res & Clin Pharm, Xuzhou 221004, Jiangsu, Peoples R ChinaGuo, Dong论文数: 0 引用数: 0 h-index: 0机构: Xuzhou Med Univ, Jiangsu Key Lab New Drug Res & Clin Pharm, Xuzhou 221004, Jiangsu, Peoples R China Xuzhou Med Univ, Jiangsu Key Lab New Drug Res & Clin Pharm, Xuzhou 221004, Jiangsu, Peoples R China
- [9] Molecular structure of a brominated 2-benzazepinone - a crucial intermediate in the synthesis of novel chemokine CCR2 receptor antagonistsZEITSCHRIFT FUR NATURFORSCHUNG SECTION B-A JOURNAL OF CHEMICAL SCIENCES, 2017, 72 (06): : 421 - 424Kokornaczyk, Artur K.论文数: 0 引用数: 0 h-index: 0机构: Wilhelms Univ Munster, Inst Pharmazeut & Med Chem Westfal, Corrensstr 48, D-48149 Munster, Germany Wilhelms Univ Munster, Inst Pharmazeut & Med Chem Westfal, Corrensstr 48, D-48149 Munster, GermanyThum, Simone论文数: 0 引用数: 0 h-index: 0机构: Wilhelms Univ Munster, Inst Pharmazeut & Med Chem Westfal, Corrensstr 48, D-48149 Munster, Germany Wilhelms Univ Munster, Inst Pharmazeut & Med Chem Westfal, Corrensstr 48, D-48149 Munster, GermanyDaniliuc, Constantin G.论文数: 0 引用数: 0 h-index: 0机构: Westfal Wilhelms Univ Munster, Organ Chem Inst, Corrensstr 40, D-48149 Munster, Germany Wilhelms Univ Munster, Inst Pharmazeut & Med Chem Westfal, Corrensstr 48, D-48149 Munster, GermanyJunker, Anna论文数: 0 引用数: 0 h-index: 0机构: Wilhelms Univ Munster, Inst Pharmazeut & Med Chem Westfal, Corrensstr 48, D-48149 Munster, Germany Westfal Wilhelms Univ, Cells Mot Cluster Excellence EXC CiM 1003, D-48149 Munster, Germany Wilhelms Univ Munster, Inst Pharmazeut & Med Chem Westfal, Corrensstr 48, D-48149 Munster, GermanyWuensch, Bernhard论文数: 0 引用数: 0 h-index: 0机构: Wilhelms Univ Munster, Inst Pharmazeut & Med Chem Westfal, Corrensstr 48, D-48149 Munster, Germany Westfal Wilhelms Univ, Cells Mot Cluster Excellence EXC CiM 1003, D-48149 Munster, Germany Wilhelms Univ Munster, Inst Pharmazeut & Med Chem Westfal, Corrensstr 48, D-48149 Munster, Germany
- [10] Synthesis and biological evaluation of spirocyclic antagonists of CCR2 (chemokine CC receptor subtype 2)BIOORGANIC & MEDICINAL CHEMISTRY, 2015, 23 (14) : 4034 - 4049Strunz, Ann Kathrin论文数: 0 引用数: 0 h-index: 0机构: Univ Munster, Inst Pharmazeut & Med Chem, D-48149 Munster, Germany Univ Munster, Inst Pharmazeut & Med Chem, D-48149 Munster, GermanyZweemer, Annelien J. M.论文数: 0 引用数: 0 h-index: 0机构: Leiden Univ, Div Med Chem, LACDR, NL-2333 CC Leiden, Netherlands Univ Munster, Inst Pharmazeut & Med Chem, D-48149 Munster, GermanyWeiss, Christina论文数: 0 引用数: 0 h-index: 0机构: Bayer Pharma AG, Global Drug Discovery Lead Discovery Wuppertal, D-42096 Wuppertal, Germany Univ Munster, Inst Pharmazeut & Med Chem, D-48149 Munster, GermanySchepmann, Dirk论文数: 0 引用数: 0 h-index: 0机构: Univ Munster, Inst Pharmazeut & Med Chem, D-48149 Munster, Germany Univ Munster, Inst Pharmazeut & Med Chem, D-48149 Munster, GermanyJunker, Anna论文数: 0 引用数: 0 h-index: 0机构: Univ Munster, Inst Pharmazeut & Med Chem, D-48149 Munster, Germany Univ Munster, Inst Pharmazeut & Med Chem, D-48149 Munster, GermanyHeitman, Laura H.论文数: 0 引用数: 0 h-index: 0机构: Leiden Univ, Div Med Chem, LACDR, NL-2333 CC Leiden, Netherlands Univ Munster, Inst Pharmazeut & Med Chem, D-48149 Munster, GermanyKoch, Michael论文数: 0 引用数: 0 h-index: 0机构: Bayer Pharma AG, Global Drug Discovery Lead Discovery Wuppertal, D-42096 Wuppertal, Germany Univ Munster, Inst Pharmazeut & Med Chem, D-48149 Munster, GermanyWuensch, Bernhard论文数: 0 引用数: 0 h-index: 0机构: Univ Munster, Inst Pharmazeut & Med Chem, D-48149 Munster, Germany Univ Munster, Cells In Mot Cluster Excellence EXC CiM 1003, D-48149 Munster, Germany Univ Munster, Inst Pharmazeut & Med Chem, D-48149 Munster, Germany