General trends in reaction of N-aryl-3-oxobutanethioamides with 2-aminoazoles(azines)

被引：5

作者：

Britsun, V. N. ^{[1
]}

Borisevich, A. N. ^{[1
]}

Lozinskii, M. O. ^{[1
]}

机构：

[1] Natl Acad Sci Ukraine, Inst Organ Chem, UA-02660 Kiev, Ukraine

来源：

RUSSIAN JOURNAL OF ORGANIC CHEMISTRY | 2007年 / 43卷 / 10期

关键词：

Pyrimidine; Thiazole; AcOH; Thione; Azine;

D O I：

10.1134/S1070428007100247

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

Reaction products obtained from N-aryl-3-oxobutanethioamides and 2-aminoazoles(azines) are derivatives of (arylamino)pyrimidines and pyrimidinethiones. The ratio of the products depends on the basicity of 1,3-binucleophiles, acidity of the medium, and the character of substituents in the phenyl ring of initial thioamides.

引用

页码：1548 / 1552

页数：5

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