A practical synthesis of nelfinavir, an HIV-protease inhibitor, using a novel chiral C4 building block:: (5R,6S)-2,2-dimethyl-5-hydroxy-1,3-dioxepan-6-ylammonium acetate

被引：37
作者：
Inaba, T
Birchler, AG
Yamada, Y
Sagawa, S
Yokota, K
Ando, K
Uchida, I
机构：
[1] Japan Tobacco Inc, Cent Pharmaceut Res Inst, Osaka 5691125, Japan
[2] Agouron Pharmaceut Inc, San Diego, CA 92121 USA
来源：
JOURNAL OF ORGANIC CHEMISTRY | 1998年 / 63卷 / 22期
关键词：
D O I：
10.1021/jo981472n
中图分类号：
O62 [有机化学];
学科分类号：
070303 ; 081704 ;
摘要：
[No abstract available]
引用
收藏
页码：7582 / 7583
页数：2
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