A one-pot, solid-phase synthesis of secondary amines from reactive alkyl halides and an alkyl azide

被引：19
|
作者：
Ayesa, Susana [1 ]
Samuelsson, Bertil [1 ]
Classon, Bjorn [1 ]
机构：
[1] Medivir AB, S-14122 Huddinge, Sweden
来源：
SYNLETT | 2008年 / 01期
关键词：
secondary amines; azides; phosphinimine; polymer-supported triphenylphosphine; alkylation;
D O I：
10.1055/s-2007-990927
中图分类号：
O62 [有机化学];
学科分类号：
070303 ; 081704 ;
摘要：
A one-pot, two-step, polymer-bound, triphenylphosphine-supported synthesis of secondary amines from the corresponding azide and a reactive alkyl halide is described.
引用
收藏
页码：97 / 99
页数：3
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