Characterization of the aggregation propensity of charge variants of recombinant human growth hormone

被引:4
作者
Meyer, Robina M. [1 ]
Aleshkevich, Sofya [1 ]
Berger, Lukas [2 ]
Nerkamp, Joerg [2 ]
Scheler, Stefan [2 ]
Friess, Wolfgang [1 ]
机构
[1] Univ Munich, Dept Pharm Pharmaceut Technol & Biopharmaceut, Butenandtstr 5, D-81377 Munich, Germany
[2] Sandoz Biopharmaceut, Biochemiestr 10, A-6336 Langkampfen, Austria
关键词
Protein charge variants; Protein aggregation; Protein stability; Temperature stress; Semi-preparative IEX; PERFORMANCE LIQUID-CHROMATOGRAPHY; PROTEIN STABILITY; IMMUNOGENICITY; ELECTROSTATICS; IDENTIFICATION; DEAMIDATION;
D O I
10.1016/j.ijpharm.2022.121760
中图分类号
R9 [药学];
学科分类号
1007 ;
摘要
Biopharmaceutical products are subject to in depth analysis to ensure and improve their safety and efficacy. As part of this effort the stability and aggregation mechanisms of the therapeutic protein is characterized over the whole life cycle. The stability and aggregation behavior of single charge variants present in biopharmaceuticals were hardly investigated. In this study we applied a previously established methodology to assess the charge variants of the drug substance (DS) of human growth hormone (hGH). We assessed the stability and aggregation propensity of an acidic variant which forms in DS at a larger extent during short time storage at elevated temperatures. We developed a semi-preparative method to separate and analyze the charge species. Thermal and colloidal stability of this variant was analyzed by light scattering methods and a stability testing in different buffer formulations. The acidic variant showed slightly attractive self-interaction at lower pH. Thermal stress did not result in increased aggregation propensity or decreased stability compared to the DS. Thus, the methodology enabled to assess the risk of a single protein variant within the DS of hGH. The approach can also be utilized for other protein drugs as previously shown for a monoclonal antibody.
引用
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页数:7
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