1,2,4-Oxadiazole ring-containing pyridylpyrazole-4-carboxamides: Synthesis and evaluation as novel insecticides of the anthranilic diamide family

被引：6

作者：

Khallaf, Abdalla ^{[1
,2
]}

Wang, Ping ^{[1
]}

Liu, Hui ^{[1
]}

Zhuo, Shuping ^{[1
]}

Zhu, Hongjun ^{[2
]}

机构：

[1] Shandong Univ Technol, Sch Chem & Chem Engn, Zibo, Peoples R China

[2] Nanjing Tech Univ, Coll Chem & Mol Engn, Dept Appl Chem, Nanjing, Peoples R China

来源：

JOURNAL OF HETEROCYCLIC CHEMISTRY | 2020年 / 57卷 / 04期

关键词：

ACTIVITY-RELATIONSHIP SAR; BIOACTIVITY; ANALOGS;

D O I：

10.1002/jhet.3927

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

Herein, we describe the preparation of pyridylpyrazole-4-carboxamides containing a 1,2,4-oxadiazole ring as novel anthranilic diamide derivatives and compare their insecticidal activities to that of chlorantraniliprole, a well-established potent insecticide. Biological activity tests reveal that all compounds had good insecticidal activities, with the most potent species achieving diamondback moth (Plutella xylostella) mortalities of 100% and 57% at concentrations of 400 and 200 mu g mL(-1), respectively.

引用

页码：1981 / 1992

页数：12

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