SYNTHESIS, BIOLOGICAL ACTIVITIES, AND TAUTOMERISM OF 4-QUINOLONES AND RELATED COMPOUNDS

被引：5

作者：

Kurasawa, Yoshihisa ^{[1
]}

Sasaki, Kenji ^{[2
,3
]}

机构：

[1] Iwaki Meisei Univ, Sch Pharm, Iwaki, Fukushima 9708551, Japan

[2] Okayama Univ, Ctr Fac Dev, Okayama 7008530, Japan

[3] Okayama Univ, Grad Sch Med Dent & Pharmaceut Sci, Kita Ku, Okayama 7008530, Japan

来源：

HETEROCYCLES | 2015年 / 91卷 / 01期

关键词：

Synthesis; Biological Activity; Tautomerism; 4-Quinolone; 4-Hydroxyquinoline; 1,3-DIPOLAR CYCLOADDITION REACTION; DIELS-ALDER REACTION; CONVENIENT SYNTHESIS; 2-SUBSTITUTED; 4-QUINOLONES; ANTIMALARIAL ACTIVITY; INHIBITORY-ACTIVITY; TOXOPLASMA-GONDII; ANALOGS; DERIVATIVES; ALKALOIDS;

D O I：

10.3987/REV-14-806

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

This review describes the synthesis, biological activities, and tautomerism of various 4-quinolones together with related compounds including 4-oxopyridazino[3,4-b]quinoxalines (bioisostere of 4-quinolones).

引用

页码：1 / 39

页数：39

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