Development of a high-throughput screening assay to identify UHRF1 inhibitors via time-resolved fluorescence resonance energy transfer (TR-FRET)

被引：2
|
作者：
Walker, David A. [1 ]
Wyhs, Nicolas [1 ]
Giovinazzo, Hugh [1 ]
Yegnasubramanian, Srinivasan [1 ]
Nelson, William G. [1 ]
机构：
[1] Johns Hopkins Sch Med, Baltimore, MD USA
来源：
CANCER RESEARCH | 2014年 / 74卷 / 19期
关键词：
D O I：
10.1158/1538-7445.AM2014-5390
中图分类号：
R73 [肿瘤学];
学科分类号：
100214 ;
摘要：
5390
引用
收藏
页数：1
相关论文
共 50 条
  • [21] Development of High-Throughput TR-FRET and AlphaScreen® Assays for Identification of Potent Inhibitors of PDK1
    Xu, Zangwei
    Nagashima, Kumiko
    Sun, Dongyu
    Rush, Thomas
    Northrup, Alan
    Andersen, Jannik N.
    Kariv, Ilona
    Bobkova, Ekaterina V.
    JOURNAL OF BIOMOLECULAR SCREENING, 2009, 14 (10) : 1257 - 1262
  • [22] Development of a time resolved FRET high-throughput assay to identify inhibitors of the RGS4/Gαo interaction
    Blazer, Levi L.
    Roman, David L.
    Neubig, Richard R.
    FASEB JOURNAL, 2007, 21 (05): : A431 - A431
  • [23] Development of a high throughput time-resolved fluorescence resonance energy transfer assay for TRAF6 ubiquitin polymerization
    Hong, CA
    Swearingen, E
    Mallari, R
    Gao, X
    Cao, ZD
    North, A
    Young, SW
    Huang, SG
    ASSAY AND DRUG DEVELOPMENT TECHNOLOGIES, 2003, 1 (01) : 175 - 180
  • [24] A 15-min non-competitive homogeneous assay for microcystin and nodularin based on time-resolved Forster resonance energy transfer (TR-FRET)
    Akter, Sultana
    Lamminmaki, Urpo
    ANALYTICAL AND BIOANALYTICAL CHEMISTRY, 2021, 413 (24) : 6159 - 6170
  • [25] A cGMP-dependent protein kinase assay for high throughput screening based on time-resolved fluorescence resonance energy transfer
    Bader, B
    Butt, E
    Palmetshofer, A
    Walter, U
    Jarchau, T
    Drueckes, P
    JOURNAL OF BIOMOLECULAR SCREENING, 2001, 6 (04) : 255 - 264
  • [26] Development of a time-resolved fluorescence resonance energy transfer ultra-high throughput screening assay targeting SYK and FCER1G interaction
    Du, Yuhong
    Wang, Dongxue
    Katis, Vittorio L.
    Zoeller, Elizabeth L.
    Qui, Min
    Levey, Allan I.
    Gileadi, Opher
    Fu, Haian
    SLAS DISCOVERY, 2024, 29 (06)
  • [27] The fluorescence resonance energy transfer (FRET) gate: A time-resolved study
    Xu, QH
    Wang, S
    Korystov, D
    Mikhailovsky, A
    Bazan, GC
    Moses, D
    Heeger, AJ
    PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA, 2005, 102 (03) : 530 - 535
  • [28] Identification of Pregnane X Receptor Ligands Using Time-Resolved Fluorescence Resonance Energy Transfer and Quantitative High-Throughput Screening
    Shukla, Sunita J.
    Nguyen, Dac-Trung
    MacArthur, Ryan
    Simeonov, Anton
    Frazee, William J.
    Hallis, Tina M.
    Marks, Bryan D.
    Singh, Upinder
    Eliason, Hildegard C.
    Printen, John
    Austin, Christopher P.
    Inglese, James
    Auld, Douglas S.
    ASSAY AND DRUG DEVELOPMENT TECHNOLOGIES, 2009, 7 (02) : 143 - 169
  • [29] A 15-min non-competitive homogeneous assay for microcystin and nodularin based on time-resolved Förster resonance energy transfer (TR-FRET)
    Sultana Akter
    Urpo Lamminmäki
    Analytical and Bioanalytical Chemistry, 2021, 413 : 6159 - 6170
  • [30] Development of a high-throughput fluorescence resonance energy transfer assay for biotin in food
    Wu, Lvliang
    Li, Yong
    Wu, Yunhua
    LWT-FOOD SCIENCE AND TECHNOLOGY, 2023, 189
12345