Discovery of pyrazolo[1,5-a]pyrimidin-7-amine derivatives as mTOR kinase domain inhibitors: Hit to lead optimization

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作者
Deng, Yongqi [1 ]
Sun, Binyuan [1 ]
Shipps, Gerald [1 ]
Matthew, Richards [1 ]
Meng, Zhaoyang [1 ]
Windsor, Williama [1 ]
Zeng, Hongbo [1 ]
Long, Brian [1 ]
Xiao, Li [1 ]
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[1] Merck Res Labs, Drug Discovery, Boston, MA 02115 USA
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O6 [化学];
学科分类号
0703 ;
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165-MEDI
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页数:1
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