Design, Synthesis and Molluscicidal Activity of New Phosphorus Compounds Bearing Fluorine Substituted 1,2,4-Triazolo[3,2-c][1,2,4]triazine Derivatives

被引:2
作者
Abdel-Rahman, Reda M. [1 ]
Alharbi, Abdulrahman S. [1 ]
Alshammari, Nawaa A. [1 ,2 ]
Adnan, Yousuf O. [1 ]
机构
[1] King Abdulaziz Univ, Fac Sci, Dept Chem, POB 42805, Jeddah 21551, Saudi Arabia
[2] Northern Borders Univ, Fac Sci, Dept Chem, Rafha, Saudi Arabia
关键词
Design; synthesis; fluorine substituted; molluscicidal; 1,2,4-triazolo[3,2-c][1,2,4]triazine; phosphorus; BIOLOGICAL EVALUATION;
D O I
10.2174/1570178616666190718120953
中图分类号
O62 [有机化学];
学科分类号
070303 ; 081704 ;
摘要
Novel phosphorus compounds bearing fluorine substituted 1,2,4-triazolo[3,2-c][1,2,4]triazine derivatives have been synthesized, starting from ring closure reactions of 3-hydrazino-4-(4'-fluoropheny1)-5-(prydin-4'-yl)-1,2,4-trizole (4) with 1,2-bioxygen compounds followed by the treatment with functional phosphorus compounds. The new systems obtained were evaluated as molluscicidal targets against some snails. Structures of these targets were elucidated upon their elemental and spectral data.
引用
收藏
页码:184 / 190
页数:7
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