Synthesis and some transformations of 2-(4-isopropyl-2-methyl-2-ethyltetrahydro-2H-pyran-4-yl)ethanamine

被引：0

作者：

Arutyunyan, N. S. ^{[1
]}

Nazaryan, R. L. ^{[1
]}

Akopyan, L. A. ^{[1
]}

Akopyan, N. Z. ^{[1
]}

Panosyan, G. A. ^{[2
]}

Gevorgyan, G. A. ^{[1
]}

机构：

[1] Natl Acad Sci Republ Armenia, Sci & Technol Ctr Organ & Pharmaceut Chem, Mnjoyan Inst Fine Organ Chem, Pr Azatutyan 26, Yerevan 0014, Armenia

[2] Natl Acad Sci Republ Armenia, Mol Struct Res Ctr, Sci & Technol Ctr Organ & Pharmaceut Chem, Yerevan, Armenia

来源：

RUSSIAN JOURNAL OF GENERAL CHEMISTRY | 2017年 / 87卷 / 07期

关键词：

acylation; reduction; decarbetoxylation; 2-(tetrahydro-2H-pyran-4-yl)ethanamine; ANTIBACTERIAL ACTIVITY; OXALATES;

D O I：

10.1134/S1070363217070313

中图分类号：

O6 [化学];

学科分类号：

0703 ;

摘要：

Condensation of 2-(4-isopropyl-2-methyl-2-ethyltetrahydro-2H-pyran-4-yl)ethanamine with aromatic aldehydes and ketones and subsequent reduction of the azomethines formed gave secondary amines of the tetrahydropyran series. Reaction of the latter with acetic acid and propionic acid chlorides provided the corresponding amides.

引用

页码：1634 / 1637

页数：4

共 5 条

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[2] SYNTHESIS AND ANTIBACTERIAL ACTIVITY OF OXALATES AND ACETAMIDES OF {2-[2-ISOPROPYLTETRAHYDROPYRAN-4-YL-4-(4-FLUOROPHENYL}ETHYL}ARYLAMINES [J].

Arutyunyan, N. S. ;

Akopyan, L. A. ;

Nazaryan, R. L. ;

Gevorgyan, G. A. ;

Stepanyan, G. M. ;

Paronikyan, R. V. ;

Panosyan, G. A. .

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[3]

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[5]

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