Recent advances in development of anthelmintic agents: Synthesis and biological screening

被引：23

作者：

Bhavsar, Zeel A. ^{[1
]}

Acharya, Prachi T. ^{[1
]}

Jethava, Divya J. ^{[1
]}

Patel, Hitesh D. ^{[1
]}

机构：

[1] Gujarat Univ, Sch Sci, Dept Chem, Ahmadabad 380009, Gujarat, India

来源：

SYNTHETIC COMMUNICATIONS | 2020年 / 50卷 / 07期

关键词：

Anthelmintic agents; biological activity; helminth infestations; heterocyclic compounds; synthesis; ONE-POT SYNTHESIS; DNA CLEAVAGE; MICROWAVE IRRADIATION; FERRITE NANOPARTICLES; MOLECULAR DOCKING; REUSABLE CATALYST; CU(II) COMPLEXES; DERIVATIVES; ANTIBACTERIAL; ANTIFUNGAL;

D O I：

10.1080/00397911.2019.1695276

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

In recent years, the use of anthelmintic agents is increased which resulted in the development of resistance to drugs. Thus, the expansion of novel anthelmintic agents is undoubtedly and most quickly escalating area in the field of medicinal chemistry. Recent research has to provide us with a significant collection of very operative and highly selective drugs, which can kill helminthic parasites efficiently. This review article describes the survey of literature regarding the variety of synthetic methods of different heterocyclic compounds and their anthelmintic activity in the last nineteen years (2001-2019). This review is primarily addressed to the description of the recent advances in the synthesis of heterocyclic compounds as anthelmintic agents, which can facilitate the development of more potent and effective anthelmintic agents.

引用

页码：917 / 946

页数：30

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