A synthesis of isocryptolepine

被引：15
作者：
Murray, PE
Mills, K
Joule, JA
机构：
[1] Univ Manchester, Dept Chem, Manchester M13 9PL, Lancs, England
[2] Glaxo Wellcome Res & Dev Ltd, Glaxo Med Res Ctr, Stevenage SG1 2NY, Herts, England
来源：
JOURNAL OF CHEMICAL RESEARCH-S | 1998年 / 07期
关键词：
D O I：
10.1039/a801313f
中图分类号：
O6 [化学];
学科分类号：
0703 ;
摘要：
A synthesis of isocryptolepine 2 is described the key steps in which are (a) palladium(o) coupling to an indol-2-ylstannane and (b) an intramolecular Vilsmeier reaction to construct the 3-aminoalkylidene-3H-indole unit of the alkaloid.
引用
收藏
页码：377 / +
页数：2
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