5(4H)-oxazolones: Synthesis and biological activities

被引:15
作者
Haneen, David S. A. [1 ]
Abou-Elmagd, Wael S. I. [1 ]
Youssef, Ahmed S. A. [1 ]
机构
[1] Ain Shams Univ, Chem Dept, Fac Sci, Cairo, Egypt
关键词
5(4H)-Oxazolones; biological evaluation; azlactones; erlenmeyer synthesis; CHLORIDE CATALYZED SYNTHESIS; ANTIBACTERIAL ACTIVITY; ANTIMICROBIAL ACTIVITY; OXAZOLONE DERIVATIVES; ACID; RING; 4-BENZYLIDENE-2-METHYL-5-OXAZOLONE; METHODOLOGY; INHIBITORS; MECHANISM;
D O I
10.1080/00397911.2020.1825746
中图分类号
O62 [有机化学];
学科分类号
070303 ; 081704 ;
摘要
In this review, we summarize all the synthetic methods and a variety of different techniques which has been used to prepare 4-arylidene-2-subsititued-5(4H)-oxazolone derivatives followed by a focused survey on the biological importance of this nucleus.
引用
收藏
页码:215 / 233
页数:19
相关论文
共 86 条
  • [1] Abdel-Aty S. A., 2009, WORLD J AGR SCI, V5
  • [2] ADAMS R, 1946, ORG REACTIONS, V3, P198
  • [3] Akram W. A. M., 2014, IJPRS, V3
  • [4] Synthesis of 4-benzylidene-oxazol-5(4H)-imines, structural analogs of PK11195, under Bischler-Napieralski conditions
    Almaraz-Giron, Marco A.
    Vazquez, Alfredo
    [J]. TETRAHEDRON LETTERS, 2017, 58 (08) : 785 - 788
  • [5] [Anonymous], 2012, INT J PHARM PHARM SC
  • [6] Microwave Assisted Improved Method for the Synthesis of Pyrazole Containing 2,4,-Disubstituted Oxazole-5-one and their Antimicrobial Activity
    Argade, N. D.
    Kalrale, B. K.
    Gill, C. H.
    [J]. E-JOURNAL OF CHEMISTRY, 2008, 5 (01) : 120 - 129
  • [7] Synthesis and antitumor activity evaluation of some novel pyrazolotriazine derivatives
    Atta-Allah, Saad R.
    Gouhar, Rasha S.
    Hemdan, Magdy M.
    Abou-Elmagd, Wael S. I.
    Haneen, David S. A.
    Kandeel, Kamal A. A.
    Youssef, Ahmed S. A.
    [J]. SYNTHETIC COMMUNICATIONS, 2017, 47 (04) : 299 - 309
  • [8] Increased microRNA-155 expression in the serum and peripheral monocytes in chronic HCV infection
    Bala, Shashi
    Tilahun, Yaphet
    Taha, Odette
    Alao, Hawau
    Kodys, Karen
    Catalano, Donna
    Szabo, Gyongyi
    [J]. JOURNAL OF TRANSLATIONAL MEDICINE, 2012, 10
  • [9] SYNTHESIS OF 2-METHYL-(Z)-4-(PHENYLIMINO)NAPHTH[2,3-D]OXAZOL-9-ONE, A MONOIMINE QUINONE WITH SELECTIVE CYTOTOXICITY TOWARD CANCER-CELLS
    BENEDETTIDOCTOROVICH, V
    BURGESS, EM
    LAMBROPOULOS, J
    LEDNICER, D
    VANDERVEER, D
    ZALKOW, LH
    [J]. JOURNAL OF MEDICINAL CHEMISTRY, 1994, 37 (05) : 710 - 712
  • [10] Bergmann M, 1926, LIEBIGS ANN CHEM, V448, P20