Synthesis and antimicrobial activity of 5-(1H-1,2,3-triazol-4-yl)-1,2,4-oxadiazole derivatives

被引：6

作者：

Krolenko, Konstantin Yu. ^{[1
]}

Vlasov, Sergiy V. ^{[1
]}

Zhuravel, Irina A. ^{[1
]}

机构：

[1] Natl Univ Pharm, 53 Pushkinska St, UA-61002 Kharkov, Ukraine

来源：

CHEMISTRY OF HETEROCYCLIC COMPOUNDS | 2016年 / 52卷 / 10期

关键词：

1,2,3-triazole; piperidine ring; pyrrolidine ring; acylation; antimicrobial activity; ANTIFUNGAL AGENTS; COMPLEXES; 1,2,3-TRIAZOLES; PALLADIUM; SAR;

D O I：

10.1007/s10593-016-1972-x

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

New 5-(1H-1,2,3-triazol-4-yl)-1,2,4-oxadiazole derivatives containing piperidine or pyrrolidine ring were synthesized and found to exhibit strong antimicrobial activity. A structure-activity study of the antimicrobial effect was performed for these compounds.

引用

页码：823 / 830

页数：8

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