Synthesis and antimicrobial activity of 5-(1H-1,2,3-triazol-4-yl)-1,2,4-oxadiazole derivatives

被引：6
|
作者：
Krolenko, Konstantin Yu. [1 ]
Vlasov, Sergiy V. [1 ]
Zhuravel, Irina A. [1 ]
机构：
[1] Natl Univ Pharm, 53 Pushkinska St, UA-61002 Kharkov, Ukraine
来源：
CHEMISTRY OF HETEROCYCLIC COMPOUNDS | 2016年 / 52卷 / 10期
关键词：
1,2,3-triazole; piperidine ring; pyrrolidine ring; acylation; antimicrobial activity; ANTIFUNGAL AGENTS; COMPLEXES; 1,2,3-TRIAZOLES; PALLADIUM; SAR;
D O I：
10.1007/s10593-016-1972-x
中图分类号：
O62 [有机化学];
学科分类号：
070303 ; 081704 ;
摘要：
New 5-(1H-1,2,3-triazol-4-yl)-1,2,4-oxadiazole derivatives containing piperidine or pyrrolidine ring were synthesized and found to exhibit strong antimicrobial activity. A structure-activity study of the antimicrobial effect was performed for these compounds.
引用
收藏
页码：823 / 830
页数：8
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