Development of an unconventional in vitro drug release test method for a bile acid sequestrant, DMP 504, tablet

被引:3
作者
Wu, LS [1 ]
McCormick, TJ [1 ]
Chang, RK [1 ]
Pang, J [1 ]
McCummings, T [1 ]
Ramos, M [1 ]
Hussain, MA [1 ]
机构
[1] Dupont Merck Pharmaceut Co, Expt Stn, Wilmington, DE 19880 USA
关键词
reverse-binding; dissolution; in vitro release; bile acid sequestrant; DMP; 504;
D O I
10.1023/A:1011916723251
中图分类号
O6 [化学];
学科分类号
0703 ;
摘要
[No abstract available]
引用
收藏
页码:1136 / 1139
页数:4
相关论文
共 6 条
[1]   INVITRO STUDIES TO INVESTIGATE THE REASONS FOR THE LOW POTENCY OF CHOLESTYRAMINE AND COLESTIPOL [J].
BENSON, GM ;
HAYNES, C ;
BLANCHARD, S ;
ELLIS, D .
JOURNAL OF PHARMACEUTICAL SCIENCES, 1993, 82 (01) :80-86
[2]  
BILLHEIMER J, 1995, 12 INT S DRUGS AFF L, V139
[3]  
GILLIES P, 1995, 12 INT S DRUGS AFF L, P139
[4]   DESCRIPTION AND SIMULATION OF A MULTIPLE MIXING TANK MODEL TO PREDICT THE EFFECT OF BILE SEQUESTRANTS ON BILE-SALT EXCRETION [J].
LUNER, PE ;
AMIDON, GL .
JOURNAL OF PHARMACEUTICAL SCIENCES, 1993, 82 (03) :311-318
[5]   EQUILIBRIUM AND KINETIC FACTORS INFLUENCING BILE SEQUESTRANT EFFICACY [J].
LUNER, PE ;
AMIDON, GL .
PHARMACEUTICAL RESEARCH, 1992, 9 (05) :670-676
[6]  
Raghavan K S, 1997, Pharm Dev Technol, V2, P233, DOI 10.3109/10837459709031443