Synthesis and Herbicidal Evaluation of Aryloxyphenoxypropionate Derivatives Containing Purine Moiety

被引：8

作者：

Shi, Jianjun ^{[1
,2
]}

Ren, Guihua ^{[1
]}

Dai, Zhimeng ^{[1
]}

Wu, Ningjie ^{[3
]}

Weng, Jianquan ^{[1
]}

Xu, Tianming ^{[3
]}

Liu, Xinghai ^{[1
]}

Tan, Chengxia ^{[1
]}

机构：

[1] Zhejiang Univ Technol, Coll Chem Engn, Hangzhou 310014, Zhejiang, Peoples R China

[2] Huangshan Univ, Sch Chem & Chem Engn, Huangshan 245041, Anhui, Peoples R China

[3] Zhejiang Res Inst Chem Ind, Natl Southern Pesticide Res Ctr, Zhejiang Base, Hangzhou 310023, Zhejiang, Peoples R China

来源：

LETTERS IN DRUG DESIGN & DISCOVERY | 2018年 / 15卷 / 01期

关键词：

Purinoxyphenoxypropionates; herbicidal activity; ACCase; synthesis; antimycobacterial; antiviral; BIOLOGICAL-ACTIVITY; ANTIFUNGAL ACTIVITY; NEMATOCIDAL ACTIVITY; BIOSYNTHESIS; INHIBITORS; SAR;

D O I：

10.2174/1570180814666170505123102

中图分类号：

R914 [药物化学];

学科分类号：

100701 ;

摘要：

Background: A series of purinoxyphenoxypropionates were designed and synthesized by introducing 8-(trifluoromethyl)-9H-purine into the aryloxyphenoxypropionate backbone. Methods: The products were characterized by H-1 NMR and HRMS. Results and Conclusion: Preliminary bioassays indicated that most of the compounds exhibited good herbicidal activity at 200 mg/L.

引用

页码：15 / 20

页数：6

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