A new and efficient synthesis of 2-aminobenzothiazoles derivatives from o-nitroaniline

被引：7
|
作者：
Mirza, Behrooz [1 ]
Mirzazadeh, Roghieh [2 ]
Zeeb, Mohsen [1 ]
机构：
[1] Islamic Azad Univ, South Tehran Branch, Fac Sci, Dept Appl Chem, Tehran, Iran
[2] Pasteur Inst Iran, Dept Biochem, Tehran, Iran
来源：
JOURNAL OF CHEMICAL RESEARCH | 2013年 / 12期
关键词：
2-aminobenzothiazoles; aryl isothiocyanates; o-nitroaniline; new precursor; IN-VIVO; AGENTS;
D O I：
10.3184/174751913X13848836801606
中图分类号：
O6 [化学];
学科分类号：
0703 ;
摘要：
A novel synthesis of 2-aminobenzothiazoles from a transition-metal-free reaction between aryl isothiocyanates and o-nitroaniline in the presence of K2CO3 is reported. The newly developed method is an efficient and cost-effective approach to synthesise 2-aminobenzothiazoles.
引用
收藏
页码：778 / 779
页数：2
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