Antifungal activity and some novel organo-phosphorus compounds: Preparation and spectral characterization

被引：3

作者：

Soni, Kusum ^{[1
]}

Jhajharia, Priyanka ^{[1
]}

Mittal, Sarita ^{[1
]}

Seth, Gita ^{[1
]}

机构：

[1] Univ Rajasthan, Dept Chem, Jaipur 302004, Rajasthan, India

来源：

PHOSPHORUS SULFUR AND SILICON AND THE RELATED ELEMENTS | 2008年 / 183卷 / 10期

关键词：

antifungal; N-phosphorylated; structure elucidation;

D O I：

10.1080/10426500801964002

中图分类号：

O61 [无机化学];

学科分类号：

070301 ; 081704 ;

摘要：

The inhibitory effects of a recently introduced series of N-phosphorylated/thiophosphorylated compounds on Aspergillus niger and Fusarium oxysporium were examined. The derivatives were obtained in good yield by reacting 2-(2'-aminophenyl)benzoxazole with phosphorous oxychloride and thiophosphoryl chloride in different molar ratios (1:1, 2:1, and 3:1). Structure elucidation of all synthesized compounds was based on the data of elemental analysis, IR, H-1 NMR, and P-31 NMR spectra.

引用

页码：2457 / 2463

页数：7

共 12 条

[1] The discovery of the potent and selective antitumour agent 2-(4-amino-3-methylphenyl)benzothiazole (DF 203) and related compounds [J].

Bradshaw, TD ;

Stevens, MFG ;

Westwell, AD .

CURRENT MEDICINAL CHEMISTRY, 2001, 8 (02) :203-210

[2] Organophosphorus derivatives containing piperazine dithiosemicarbazones as chemotherapeutants against fungal pathogens of sugarcane [J].

Chandra, R ;

Pandey, OP ;

Sengupta, SK .

JOURNAL OF AGRICULTURAL AND FOOD CHEMISTRY, 2005, 53 (06) :2181-2184

[3] Antitumor benzothiazoles. 7. Synthesis of 2-(4-acylaminophenyl)benzothiazoles and investigations into the role of acetylation in the antitumor activities of the parent amines [J].

Chua, MS ;

Shi, DF ;

Wrigley, S ;

Bradshaw, TD ;

Hutchinson, I ;

Shaw, PN ;

Barrett, DA ;

Stanley, LA ;

Stevens, MFG .

JOURNAL OF MEDICINAL CHEMISTRY, 1999, 42 (03) :381-392

[4] One-pot synthesis and fungicidal activity of pyrimidinylidenamido- and thiazolinylidenamidomonothiophosphoric esters [J].

Gupta, N ;

Kabra, V ;

Saxena, V ;

Jain, S ;

Bhatnager, K .

PHOSPHORUS SULFUR AND SILICON AND THE RELATED ELEMENTS, 2003, 178 (04) :851-861

[5]

John PJ, 2000, TRIBOL LETT, V9, P167

[6]

Karali N, 2004, INDIAN J CHEM B, V43, P212

[7] A stepwise one pot synthesis of alkyl thiophosphoramidate derivatives of nucleosides [J].

Miao, ZW ;

Fu, H ;

Han, B ;

Chen, Y ;

Zhao, YF .

SYNTHETIC COMMUNICATIONS, 2002, 32 (08) :1159-1167

[8] Synthesis and bioassay of phosphorylated and thiophosphorylated derivatives of substituted benzothiazoles [J].

Mittal, S. ;

Samota, M. K. ;

Kaur, J. ;

Seth, Gita .

PHOSPHORUS SULFUR AND SILICON AND THE RELATED ELEMENTS, 2006, 181 (12) :2843-2849

[9] Synthesis and antibacterial activity of new 2-aryloxy-6-bromo-3-(4-chlorophenyl)-3,4-dihydrobenzo[e][1,3,2]oxazaphosphinine 2-oxides [J].

Prasad, Gandavaram Syam ;

Babu, Boppudi Hari ;

Reddy, Kachi Kishore Kumar Reddy ;

Haranath, Pallam Reddy ;

Reddy, Cirandur Suresh .

ARKIVOC, 2006, :165-170

[10] Synthesis and biological activity of some novel O-phosphorylated benzoxazole derivatives [J].

Samota, M. K. ;

Kumar, A. ;

Kaur, J. ;

Mittal, S. ;

Seth, Gita .

PHOSPHORUS SULFUR AND SILICON AND THE RELATED ELEMENTS, 2006, 181 (08) :1919-1924

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