Synthesis of a [1,4]dioxane-2,5-dione based-peptidomimetic scaffold

被引：0
|
作者：
Abell, Andrew D. [1 ]
Harvey, Andrew J. [1 ]
机构：
[1] Univ Canterbury, Dept Chem, Christchurch 1, New Zealand
来源：
ARKIVOC | 2006年
关键词：
peptidomimetic scaffold; synthesis; dimer; cyclisation;
D O I：
暂无
中图分类号：
O62 [有机化学];
学科分类号：
070303 ; 081704 ;
摘要：
(2S,3S)-3-[N-Cbz-L-Leucinyl]amino-2-hydroxy-4-phenylbutanoic acid 5 dimerised on treatment with EDCI and HOBT to give the symmetrical [1,4]dioxane-2,5-dione-based peptidomimetic 6.
引用
收藏
页码：72 / 76
页数：5
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