Expeditious synthesis of novel NK1 antagonists based on a 1,2,4-trisubstituted cyclohexane

被引：8

作者：

Dirat, O ^{[1
]}

Elliott, JM ^{[1
]}

Jelley, RA ^{[1
]}

Jones, AB ^{[1
]}

Reader, M ^{[1
]}

机构：

[1] Merck Sharp & Dohme Res Labs, Ctr Res Neurosci, Dept Med Chem, Harlow CM20 2QR, Essex, England

来源：

TETRAHEDRON LETTERS | 2006年 / 47卷 / 08期

关键词：

NK1; asymmetric synthesis; triazole; alpha-arylation;

D O I：

10.1016/j.tetlet.2005.12.067

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

引用

页码：1295 / 1298

页数：4

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