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- [1] Clinical activity of LY2835219, a novel cell cycle inhibitor selective for CDK4 and CDK6, in patients with metastatic breast cancerCANCER RESEARCH, 2014, 74 (19)Patnaik, Amita论文数: 0 引用数: 0 h-index: 0机构: START, San Antonio, TX USA START, San Antonio, TX USARosen, Lee S.论文数: 0 引用数: 0 h-index: 0机构: Univ Calif Los Angeles, Santa Monica, CA USA START, San Antonio, TX USATolaney, Sara M.论文数: 0 引用数: 0 h-index: 0机构: Dana Farber Canc Inst, Boston, MA 02115 USA START, San Antonio, TX USATolcher, Anthony W.论文数: 0 引用数: 0 h-index: 0机构: START, San Antonio, TX USA START, San Antonio, TX USAGoldman, Jonathan W.论文数: 0 引用数: 0 h-index: 0机构: Univ Calif Los Angeles, Santa Monica, CA USA START, San Antonio, TX USA论文数: 引用数: h-index:机构:Papadopoulos, Kyriakos P.论文数: 0 引用数: 0 h-index: 0机构: START, San Antonio, TX USA START, San Antonio, TX USABeeram, Muralidhar论文数: 0 引用数: 0 h-index: 0机构: START, San Antonio, TX USA START, San Antonio, TX USARasco, Drew W.论文数: 0 引用数: 0 h-index: 0机构: START, San Antonio, TX USA START, San Antonio, TX USAMyrand, Scott P.论文数: 0 引用数: 0 h-index: 0机构: Eli Lilly & Co, Indianapolis, IN 46285 USA START, San Antonio, TX USAKulanthaivel, Palaniappan论文数: 0 引用数: 0 h-index: 0机构: Eli Lilly & Co, Indianapolis, IN 46285 USA START, San Antonio, TX USALi, Lily论文数: 0 引用数: 0 h-index: 0机构: Eli Lilly & Co, Indianapolis, IN 46285 USA START, San Antonio, TX USAFrenzel, Martin论文数: 0 引用数: 0 h-index: 0机构: Eli Lilly & Co, Indianapolis, IN 46285 USA START, San Antonio, TX USACronier, Damien M.论文数: 0 引用数: 0 h-index: 0机构: Eli Lilly & Co, Indianapolis, IN 46285 USA START, San Antonio, TX USAChan, Edward M.论文数: 0 引用数: 0 h-index: 0机构: Eli Lilly & Co, Indianapolis, IN 46285 USA START, San Antonio, TX USAFlaherty, Keith T.论文数: 0 引用数: 0 h-index: 0机构: Massachusetts Gen Hosp, Ctr Canc, Boston, MA USA START, San Antonio, TX USAWen, Patrick Y.论文数: 0 引用数: 0 h-index: 0机构: Dana Farber Canc Inst, Boston, MA 02115 USA START, San Antonio, TX USAShapiro, Geoffrey I.论文数: 0 引用数: 0 h-index: 0机构: Dana Farber Canc Inst, Boston, MA 02115 USA START, San Antonio, TX USA
- [2] Clinical activity of LY2835219, a novel cell cycle inhibitor selective for CDK4 and CDK6, in patients with non-small cell lung cancer.JOURNAL OF CLINICAL ONCOLOGY, 2014, 32 (15)Goldman, Jonathan Wade论文数: 0 引用数: 0 h-index: 0机构: Univ Calif Los Angeles, Santa Monica Hematol Oncol, Santa Monica, CA USAGandhi, Leena论文数: 0 引用数: 0 h-index: 0机构: Univ Calif Los Angeles, Santa Monica Hematol Oncol, Santa Monica, CA USAPatnaik, Amita论文数: 0 引用数: 0 h-index: 0机构: Univ Calif Los Angeles, Santa Monica Hematol Oncol, Santa Monica, CA USARosen, Lee S.论文数: 0 引用数: 0 h-index: 0机构: Univ Calif Los Angeles, Santa Monica Hematol Oncol, Santa Monica, CA USAHilton, John Frederick论文数: 0 引用数: 0 h-index: 0机构: Univ Calif Los Angeles, Santa Monica Hematol Oncol, Santa Monica, CA USAPapadopoulos, Kyriakos P.论文数: 0 引用数: 0 h-index: 0机构: Univ Calif Los Angeles, Santa Monica Hematol Oncol, Santa Monica, CA USATolaney, Sara M.论文数: 0 引用数: 0 h-index: 0机构: Univ Calif Los Angeles, Santa Monica Hematol Oncol, Santa Monica, CA USABeeram, Muralidhar论文数: 0 引用数: 0 h-index: 0机构: Univ Calif Los Angeles, Santa Monica Hematol Oncol, Santa Monica, CA USARasco, Drew Warren论文数: 0 引用数: 0 h-index: 0机构: Univ Calif Los Angeles, Santa Monica Hematol Oncol, Santa Monica, CA USAMyrand, Scott P.论文数: 0 引用数: 0 h-index: 0机构: Univ Calif Los Angeles, Santa Monica Hematol Oncol, Santa Monica, CA USABeckmann, Richard P.论文数: 0 引用数: 0 h-index: 0机构: Univ Calif Los Angeles, Santa Monica Hematol Oncol, Santa Monica, CA USAKulanthaivel, Palaniappan论文数: 0 引用数: 0 h-index: 0机构: Univ Calif Los Angeles, Santa Monica Hematol Oncol, Santa Monica, CA USAFrenzel, Martin论文数: 0 引用数: 0 h-index: 0机构: Univ Calif Los Angeles, Santa Monica Hematol Oncol, Santa Monica, CA USACronier, Damien论文数: 0 引用数: 0 h-index: 0机构: Univ Calif Los Angeles, Santa Monica Hematol Oncol, Santa Monica, CA USAChan, Edward M.论文数: 0 引用数: 0 h-index: 0机构: Univ Calif Los Angeles, Santa Monica Hematol Oncol, Santa Monica, CA USAFlaherty, Keith论文数: 0 引用数: 0 h-index: 0机构: Univ Calif Los Angeles, Santa Monica Hematol Oncol, Santa Monica, CA USAWen, Patrick Y.论文数: 0 引用数: 0 h-index: 0机构: Univ Calif Los Angeles, Santa Monica Hematol Oncol, Santa Monica, CA USATolcher, Anthony W.论文数: 0 引用数: 0 h-index: 0机构: Univ Calif Los Angeles, Santa Monica Hematol Oncol, Santa Monica, CA USAShapiro, Geoffrey论文数: 0 引用数: 0 h-index: 0机构: Univ Calif Los Angeles, Santa Monica Hematol Oncol, Santa Monica, CA USA
- [3] A first-in-human phase I study of the CDK4/6 inhibitor, LY2835219, for patients with advanced cancer.JOURNAL OF CLINICAL ONCOLOGY, 2013, 31 (15)Shapiro, Geoffrey论文数: 0 引用数: 0 h-index: 0机构: Dana Farber Canc Inst, Boston, MA 02115 USARosen, Lee S.论文数: 0 引用数: 0 h-index: 0机构: Dana Farber Canc Inst, Boston, MA 02115 USATolcher, Anthony W.论文数: 0 引用数: 0 h-index: 0机构: Dana Farber Canc Inst, Boston, MA 02115 USAGoldman, Jonathan Wade论文数: 0 引用数: 0 h-index: 0机构: Dana Farber Canc Inst, Boston, MA 02115 USAGandhi, Leena论文数: 0 引用数: 0 h-index: 0机构: Dana Farber Canc Inst, Boston, MA 02115 USAPapadopoulos, Kyriakos P.论文数: 0 引用数: 0 h-index: 0机构: Dana Farber Canc Inst, Boston, MA 02115 USATolaney, Sara M.论文数: 0 引用数: 0 h-index: 0机构: Dana Farber Canc Inst, Boston, MA 02115 USABeeram, Muralidhar论文数: 0 引用数: 0 h-index: 0机构: Dana Farber Canc Inst, Boston, MA 02115 USARasco, Drew Warren论文数: 0 引用数: 0 h-index: 0机构: Dana Farber Canc Inst, Boston, MA 02115 USAKulanthaivel, Palaniappan论文数: 0 引用数: 0 h-index: 0机构: Dana Farber Canc Inst, Boston, MA 02115 USALi, Qian论文数: 0 引用数: 0 h-index: 0机构: Dana Farber Canc Inst, Boston, MA 02115 USAHu, Tianle论文数: 0 引用数: 0 h-index: 0机构: Dana Farber Canc Inst, Boston, MA 02115 USACronier, Damien论文数: 0 引用数: 0 h-index: 0机构: Dana Farber Canc Inst, Boston, MA 02115 USAChan, Edward M.论文数: 0 引用数: 0 h-index: 0机构: Dana Farber Canc Inst, Boston, MA 02115 USAFlaherty, Keith论文数: 0 引用数: 0 h-index: 0机构: Dana Farber Canc Inst, Boston, MA 02115 USAWen, Patrick Y.论文数: 0 引用数: 0 h-index: 0机构: Dana Farber Canc Inst, Boston, MA 02115 USAPatnaik, Amita论文数: 0 引用数: 0 h-index: 0机构: Dana Farber Canc Inst, Boston, MA 02115 USA
- [4] Clinical Activity of Abemaciclib (LY2835219), a Cell Cycle Inhibitor Selective for CDK4 and CDK6, in Patients with Relapsed or Refractory Mantle Cell LymphomaBLOOD, 2014, 124 (21)Morschhauser, Franck论文数: 0 引用数: 0 h-index: 0机构: CHRU Lille, Hop Claude Huriez, F-59037 Lille, France CHRU Lille, Hop Claude Huriez, F-59037 Lille, FranceBouabdallah, Kamal论文数: 0 引用数: 0 h-index: 0机构: Hop Haut Leveque, Pessac, France CHRU Lille, Hop Claude Huriez, F-59037 Lille, FranceStilgenbauer, Stephan论文数: 0 引用数: 0 h-index: 0机构: Univ Ulm, D-89069 Ulm, Germany CHRU Lille, Hop Claude Huriez, F-59037 Lille, FranceThieblemont, Catherine论文数: 0 引用数: 0 h-index: 0机构: Hop St Louis, Paris, France CHRU Lille, Hop Claude Huriez, F-59037 Lille, FranceWolf, Martin论文数: 0 引用数: 0 h-index: 0机构: Klinikum Kassel, Kassel, Germany CHRU Lille, Hop Claude Huriez, F-59037 Lille, Francede Guibert, Sophie论文数: 0 引用数: 0 h-index: 0机构: Univ Hosp, Rennes, France CHRU Lille, Hop Claude Huriez, F-59037 Lille, FranceZettl, Florian论文数: 0 引用数: 0 h-index: 0机构: Univ Hosp, Gottingen, Germany CHRU Lille, Hop Claude Huriez, F-59037 Lille, FranceHahka-Kemppinen, Marjo论文数: 0 引用数: 0 h-index: 0机构: Eli Lilly & Co, Helsinki, Finland CHRU Lille, Hop Claude Huriez, F-59037 Lille, FranceWang, David Xiaohui论文数: 0 引用数: 0 h-index: 0机构: Eli Lilly & Co, Neuilly Sur Seine, France CHRU Lille, Hop Claude Huriez, F-59037 Lille, FranceBrueck, Patrick论文数: 0 引用数: 0 h-index: 0机构: Eli Lilly & Co, Bad Homburg, Germany CHRU Lille, Hop Claude Huriez, F-59037 Lille, FranceCaldwell, Charles论文数: 0 引用数: 0 h-index: 0机构: Eli Lilly & Co, Indianapolis, IN 46285 USA CHRU Lille, Hop Claude Huriez, F-59037 Lille, FranceBeckmann, Richard论文数: 0 引用数: 0 h-index: 0机构: Eli Lilly & Co, Indianapolis, IN 46285 USA CHRU Lille, Hop Claude Huriez, F-59037 Lille, FranceGelbert, Lawrence论文数: 0 引用数: 0 h-index: 0机构: Indiana Univ Sch Med, Indianapolis, IN 46202 USA CHRU Lille, Hop Claude Huriez, F-59037 Lille, FranceCronier, Damien论文数: 0 引用数: 0 h-index: 0机构: Eli Lilly & Co, Windlesham, Surrey, England CHRU Lille, Hop Claude Huriez, F-59037 Lille, FranceLin, Ji论文数: 0 引用数: 0 h-index: 0机构: Eli Lilly & Co, Indianapolis, IN 46285 USA CHRU Lille, Hop Claude Huriez, F-59037 Lille, FranceLi, Lily论文数: 0 引用数: 0 h-index: 0机构: Eli Lilly & Co, Indianapolis, IN 46285 USA CHRU Lille, Hop Claude Huriez, F-59037 Lille, FranceChan, Edward M.论文数: 0 引用数: 0 h-index: 0机构: Eli Lilly & Co, Indianapolis, IN 46285 USA CHRU Lille, Hop Claude Huriez, F-59037 Lille, FrancePfreundschuh, Michael论文数: 0 引用数: 0 h-index: 0机构: Univ Hosp Saarland, Homburg, Germany CHRU Lille, Hop Claude Huriez, F-59037 Lille, FranceWilhem, Martin论文数: 0 引用数: 0 h-index: 0机构: Klinikum Nuernberg Nord, Nurnberg, Germany CHRU Lille, Hop Claude Huriez, F-59037 Lille, FranceHess, Georg论文数: 0 引用数: 0 h-index: 0机构: Univ Med Mainz, Mainz, Germany CHRU Lille, Hop Claude Huriez, F-59037 Lille, France
- [5] LY2835219, a novel cell cycle inhibitor selective for CDK4/6, in combination with fulvestrant for patients with hormone receptor positive (HR plus ) metastatic breast cancer.JOURNAL OF CLINICAL ONCOLOGY, 2014, 32 (15)Patnaik, Amita论文数: 0 引用数: 0 h-index: 0机构: South Texas Accelerated Res Therapeut START Ctr C, San Antonio, TX USARosen, Lee S.论文数: 0 引用数: 0 h-index: 0机构: South Texas Accelerated Res Therapeut START Ctr C, San Antonio, TX USATolaney, Sara M.论文数: 0 引用数: 0 h-index: 0机构: South Texas Accelerated Res Therapeut START Ctr C, San Antonio, TX USATolcher, Anthony W.论文数: 0 引用数: 0 h-index: 0机构: South Texas Accelerated Res Therapeut START Ctr C, San Antonio, TX USAGoldman, Jonathan Wade论文数: 0 引用数: 0 h-index: 0机构: South Texas Accelerated Res Therapeut START Ctr C, San Antonio, TX USAGandhi, Leena论文数: 0 引用数: 0 h-index: 0机构: South Texas Accelerated Res Therapeut START Ctr C, San Antonio, TX USAPapadopoulos, Kyriakos P.论文数: 0 引用数: 0 h-index: 0机构: South Texas Accelerated Res Therapeut START Ctr C, San Antonio, TX USABeeram, Muralidhar论文数: 0 引用数: 0 h-index: 0机构: South Texas Accelerated Res Therapeut START Ctr C, San Antonio, TX USARasco, Drew Warren论文数: 0 引用数: 0 h-index: 0机构: South Texas Accelerated Res Therapeut START Ctr C, San Antonio, TX USAMyrand, Scott P.论文数: 0 引用数: 0 h-index: 0机构: South Texas Accelerated Res Therapeut START Ctr C, San Antonio, TX USAKulanthaivel, Palaniappan论文数: 0 引用数: 0 h-index: 0机构: South Texas Accelerated Res Therapeut START Ctr C, San Antonio, TX USAAndrews, Joan M.论文数: 0 引用数: 0 h-index: 0机构: South Texas Accelerated Res Therapeut START Ctr C, San Antonio, TX USAFrenzel, Martin论文数: 0 引用数: 0 h-index: 0机构: South Texas Accelerated Res Therapeut START Ctr C, San Antonio, TX USACronier, Damien论文数: 0 引用数: 0 h-index: 0机构: South Texas Accelerated Res Therapeut START Ctr C, San Antonio, TX USAChan, Edward M.论文数: 0 引用数: 0 h-index: 0机构: South Texas Accelerated Res Therapeut START Ctr C, San Antonio, TX USAFlaherty, Keith论文数: 0 引用数: 0 h-index: 0机构: South Texas Accelerated Res Therapeut START Ctr C, San Antonio, TX USAWen, Patrick Y.论文数: 0 引用数: 0 h-index: 0机构: South Texas Accelerated Res Therapeut START Ctr C, San Antonio, TX USAShapiro, Geoffrey论文数: 0 引用数: 0 h-index: 0机构: South Texas Accelerated Res Therapeut START Ctr C, San Antonio, TX USA
- [6] Combination of CDK4/6 inhibitor, LY2835219, and mTOR inhibitor to synergistically suppress the growth of head and neck squamous cell carcinomaJOURNAL OF CLINICAL ONCOLOGY, 2016, 34 (15)Ahn, Myung-Ju论文数: 0 引用数: 0 h-index: 0机构: Sungkyunkwan Univ, Div Hematol & Oncol, Dept Med, Samsung Med Ctr,Sch Med, Seoul, South KoreaKu, Bo Mi论文数: 0 引用数: 0 h-index: 0机构: Sungkyunkwan Univ, Div Hematol & Oncol, Dept Med, Samsung Med Ctr,Sch Med, Seoul, South KoreaYi, Seong Yoon论文数: 0 引用数: 0 h-index: 0机构: Sungkyunkwan Univ, Div Hematol & Oncol, Dept Med, Samsung Med Ctr,Sch Med, Seoul, South KoreaKoh, Jiae论文数: 0 引用数: 0 h-index: 0机构: Sungkyunkwan Univ, Div Hematol & Oncol, Dept Med, Samsung Med Ctr,Sch Med, Seoul, South KoreaBae, Yeon-Hee论文数: 0 引用数: 0 h-index: 0机构: Sungkyunkwan Univ, Div Hematol & Oncol, Dept Med, Samsung Med Ctr,Sch Med, Seoul, South KoreaSun, Jong-Mu论文数: 0 引用数: 0 h-index: 0机构: Sungkyunkwan Univ, Div Hematol & Oncol, Dept Med, Samsung Med Ctr,Sch Med, Seoul, South KoreaLee, Se-Hoon论文数: 0 引用数: 0 h-index: 0机构: Sungkyunkwan Univ, Div Hematol & Oncol, Dept Med, Samsung Med Ctr,Sch Med, Seoul, South KoreaAhn, Jin Seok论文数: 0 引用数: 0 h-index: 0机构: Sungkyunkwan Univ, Div Hematol & Oncol, Dept Med, Samsung Med Ctr,Sch Med, Seoul, South KoreaPark, Keunchil论文数: 0 引用数: 0 h-index: 0机构: Sungkyunkwan Univ, Div Hematol & Oncol, Dept Med, Samsung Med Ctr,Sch Med, Seoul, South Korea
- [7] CDK4/6 inhibitor (LY2835219) exhibits potent anti-tumor activity in human lung cancer cell lines with intact retinoblastomaEUROPEAN JOURNAL OF CANCER, 2014, 50 : 162 - 162Goldman, J. W.论文数: 0 引用数: 0 h-index: 0机构: Univ Calif Los Angeles, David Geffen Sch Med, Dept Med, Div Hematol Oncol, Los Angeles, CA 90095 USA Univ Calif Los Angeles, David Geffen Sch Med, Dept Med, Div Hematol Oncol, Los Angeles, CA 90095 USAGaron, E. B.论文数: 0 引用数: 0 h-index: 0机构: Univ Calif Los Angeles, David Geffen Sch Med, Dept Med, Div Hematol Oncol, Los Angeles, CA 90095 USA Univ Calif Los Angeles, David Geffen Sch Med, Dept Med, Div Hematol Oncol, Los Angeles, CA 90095 USAConklin, D.论文数: 0 引用数: 0 h-index: 0机构: Univ Calif Los Angeles, David Geffen Sch Med, Dept Med, Div Hematol Oncol, Los Angeles, CA 90095 USA Univ Calif Los Angeles, David Geffen Sch Med, Dept Med, Div Hematol Oncol, Los Angeles, CA 90095 USAWong, D. J. L.论文数: 0 引用数: 0 h-index: 0机构: Univ Calif Los Angeles, David Geffen Sch Med, Dept Med, Div Hematol Oncol, Los Angeles, CA 90095 USA Univ Calif Los Angeles, David Geffen Sch Med, Dept Med, Div Hematol Oncol, Los Angeles, CA 90095 USAWolf, B.论文数: 0 引用数: 0 h-index: 0机构: Univ Calif Los Angeles, David Geffen Sch Med, Dept Med, Div Hematol Oncol, Los Angeles, CA 90095 USA Univ Calif Los Angeles, David Geffen Sch Med, Dept Med, Div Hematol Oncol, Los Angeles, CA 90095 USASilveira, D. D.论文数: 0 引用数: 0 h-index: 0机构: Univ Calif Los Angeles, David Geffen Sch Med, Dept Med, Div Hematol Oncol, Los Angeles, CA 90095 USA Univ Calif Los Angeles, David Geffen Sch Med, Dept Med, Div Hematol Oncol, Los Angeles, CA 90095 USAKamranpour, N.论文数: 0 引用数: 0 h-index: 0机构: Univ Calif Los Angeles, David Geffen Sch Med, Dept Med, Div Hematol Oncol, Los Angeles, CA 90095 USA Univ Calif Los Angeles, David Geffen Sch Med, Dept Med, Div Hematol Oncol, Los Angeles, CA 90095 USAPitts, S.论文数: 0 引用数: 0 h-index: 0机构: Univ Calif Los Angeles, David Geffen Sch Med, Dept Med, Div Hematol Oncol, Los Angeles, CA 90095 USA Univ Calif Los Angeles, David Geffen Sch Med, Dept Med, Div Hematol Oncol, Los Angeles, CA 90095 USAFinn, R. S.论文数: 0 引用数: 0 h-index: 0机构: Univ Calif Los Angeles, David Geffen Sch Med, Dept Med, Div Hematol Oncol, Los Angeles, CA 90095 USA Univ Calif Los Angeles, David Geffen Sch Med, Dept Med, Div Hematol Oncol, Los Angeles, CA 90095 USASlamon, D. J.论文数: 0 引用数: 0 h-index: 0机构: Univ Calif Los Angeles, David Geffen Sch Med, Dept Med, Div Hematol Oncol, Los Angeles, CA 90095 USA Univ Calif Los Angeles, David Geffen Sch Med, Dept Med, Div Hematol Oncol, Los Angeles, CA 90095 USA
- [8] Preclinical head-to-head comparison of CDK4/6 inhibitor activity toward CDK4 vs CDK6CANCER RESEARCH, 2021, 81 (04)Delach, Scott论文数: 0 引用数: 0 h-index: 0机构: Novartis Inst Biomed Res, Cambridge, MA USA Novartis Inst Biomed Res, Cambridge, MA USACaponigro, Giordano论文数: 0 引用数: 0 h-index: 0机构: Novartis Inst Biomed Res, Cambridge, MA USA Novartis Inst Biomed Res, Cambridge, MA USA
- [9] Targeting CDK4 and CDK6 in cancerNature Reviews Cancer, 2022, 22 : 356 - 372Shom Goel论文数: 0 引用数: 0 h-index: 0机构: Peter MacCallum Cancer Centre,Sir Peter MacCallum Department of OncologyJohann S. Bergholz论文数: 0 引用数: 0 h-index: 0机构: Peter MacCallum Cancer Centre,Sir Peter MacCallum Department of OncologyJean J. Zhao论文数: 0 引用数: 0 h-index: 0机构: Peter MacCallum Cancer Centre,Sir Peter MacCallum Department of Oncology
- [10] Targeting CDK4 and CDK6 in cancerNATURE REVIEWS CANCER, 2022, 22 (06) : 356 - 372论文数: 引用数: h-index:机构:Bergholz, Johann S.论文数: 0 引用数: 0 h-index: 0机构: Dana Farber Canc Inst, Boston, MA 02115 USA Harvard Med Sch, Boston, MA 02115 USA Broad Inst Harvard & MIT, Cambridge, MA 02142 USA Peter MacCallum Canc Ctr, Melbourne, Vic, AustraliaZhao, Jean J.论文数: 0 引用数: 0 h-index: 0机构: Dana Farber Canc Inst, Boston, MA 02115 USA Harvard Med Sch, Boston, MA 02115 USA Broad Inst Harvard & MIT, Cambridge, MA 02142 USA Peter MacCallum Canc Ctr, Melbourne, Vic, Australia