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- [1] Safety and efficacy of oral JAK inhibitors PF-06651600 and PF-06700841 in a withdrawal/retreatment study in patients with alopecia areataAUSTRALASIAN JOURNAL OF DERMATOLOGY, 2021, 62 : 116 - 117Peeva, E.论文数: 0 引用数: 0 h-index: 0机构: Pfizer, Cambridge, MA USA Pfizer, Cambridge, MA USABanerjee, A.论文数: 0 引用数: 0 h-index: 0机构: Pfizer, Cambridge, MA USA Pfizer, Cambridge, MA USAGuttman-Yassky, E.论文数: 0 引用数: 0 h-index: 0机构: Icahn Sch Med Mt Sinai, New York, NY 10029 USA Pfizer, Cambridge, MA USASinclair, R.论文数: 0 引用数: 0 h-index: 0机构: Sinclair Dermatol, Melbourne, Vic, Australia Pfizer, Cambridge, MA USACox, L. A.论文数: 0 引用数: 0 h-index: 0机构: Pfizer, Cambridge, MA USA Pfizer, Cambridge, MA USAZhu, L.论文数: 0 引用数: 0 h-index: 0机构: Pfizer, Cambridge, MA USA Pfizer, Cambridge, MA USAZhu, H.论文数: 0 引用数: 0 h-index: 0机构: Pfizer, Shanghai, Peoples R China Pfizer, Cambridge, MA USAVincent, M.论文数: 0 引用数: 0 h-index: 0机构: Pfizer, Cambridge, MA USA Pfizer, Cambridge, MA USAKing, B.论文数: 0 引用数: 0 h-index: 0机构: Yale Univ, Sch Med, New Haven, CT USA Pfizer, Cambridge, MA USA
- [2] Evaluation of pharmacology and clinical response to TYK2/JAK1 kinase inhibitor, PF-06700841, in patients with plaque psoriasisJOURNAL OF THE AMERICAN ACADEMY OF DERMATOLOGY, 2017, 76 (06) : AB130 - AB130Page, Karen M.论文数: 0 引用数: 0 h-index: 0机构: Pfizer, New York, NY USA Pfizer, New York, NY USAZhang, Weidong论文数: 0 引用数: 0 h-index: 0机构: Pfizer, New York, NY USA Pfizer, New York, NY USAScaramozza, Matthew论文数: 0 引用数: 0 h-index: 0机构: Pfizer, New York, NY USA Pfizer, New York, NY USASuprun, Maria论文数: 0 引用数: 0 h-index: 0机构: Icahn Sch Med Mt Sinai, New York, NY 10029 USA Pfizer, New York, NY USASuarez-Farinas, Mayte论文数: 0 引用数: 0 h-index: 0机构: Icahn Sch Med Mt Sinai, New York, NY 10029 USA Pfizer, New York, NY USAFuentes-Duculan, Judilyn论文数: 0 引用数: 0 h-index: 0机构: Rockefeller Univ, 1230 York Ave, New York, NY 10021 USA Pfizer, New York, NY USAJames, G. Krueger论文数: 0 引用数: 0 h-index: 0机构: Rockefeller Univ, 1230 York Ave, New York, NY 10021 USA Pfizer, New York, NY USAWinkle, Peter J.论文数: 0 引用数: 0 h-index: 0机构: Anaheim Clin Trials, Anaheim, CA USA Pfizer, New York, NY USAPeeva, Elena论文数: 0 引用数: 0 h-index: 0机构: Pfizer, New York, NY USA Pfizer, New York, NY USA
- [3] Clinical efficacy of the oral JAK3/TEC inhibitor ritlecitinib (PF-06651600) and patients' perception of improvement in alopecia areata: Results from the ALLEGRO Phase 2b/3 trialEXPERIMENTAL DERMATOLOGY, 2021, 30 : 20 - 20Guttman-Yassky, E.论文数: 0 引用数: 0 h-index: 0机构: Icahn Sch Med Mt Sinai, New York, NY 10029 USA Icahn Sch Med Mt Sinai, New York, NY 10029 USAIto, T.论文数: 0 引用数: 0 h-index: 0机构: Hamamatsu Univ Sch Med, Dept Dermatol, Hamamatsu, Shizuoka, Japan Icahn Sch Med Mt Sinai, New York, NY 10029 USAJabbari, A.论文数: 0 引用数: 0 h-index: 0机构: Univ Iowa, Dept Dermatol, Iowa City, IA 52242 USA Icahn Sch Med Mt Sinai, New York, NY 10029 USAMackay-Wiggan, J.论文数: 0 引用数: 0 h-index: 0机构: Siperstein Dermatol Grp, Boynton Beach, FL USA Icahn Sch Med Mt Sinai, New York, NY 10029 USALejeune, A.论文数: 0 引用数: 0 h-index: 0机构: Pfizer, Paris, France Icahn Sch Med Mt Sinai, New York, NY 10029 USAWolk, R.论文数: 0 引用数: 0 h-index: 0机构: Pfizer, Groton, CT USA Icahn Sch Med Mt Sinai, New York, NY 10029 USAWajsbrot, D.论文数: 0 引用数: 0 h-index: 0机构: Pfizer, New York, NY USA Icahn Sch Med Mt Sinai, New York, NY 10029 USAZwillich, S. H.论文数: 0 引用数: 0 h-index: 0机构: Pfizer, Groton, CT USA Icahn Sch Med Mt Sinai, New York, NY 10029 USA
- [4] Selective oral JAK3 and TYK2/JAK1 kinase inhibitors both demonstrate significant hair-growth compared to placebo and improvement of hair-associated keratins in patients with moderate-to-severe Alopecia AreataEXPERIMENTAL DERMATOLOGY, 2018, 27 : 52 - 53Guttman-Yassky, E.论文数: 0 引用数: 0 h-index: 0机构: Icahn Sch Med Mt Sinai, New York, NY 10029 USA Icahn Sch Med Mt Sinai, New York, NY 10029 USAPage, K.论文数: 0 引用数: 0 h-index: 0机构: Pfizer Inc, Cambridge, England Icahn Sch Med Mt Sinai, New York, NY 10029 USAPavel, A. B.论文数: 0 引用数: 0 h-index: 0机构: Icahn Sch Med Mt Sinai, New York, NY 10029 USA Icahn Sch Med Mt Sinai, New York, NY 10029 USADiaz, A.论文数: 0 引用数: 0 h-index: 0机构: Icahn Sch Med Mt Sinai, New York, NY 10029 USA Icahn Sch Med Mt Sinai, New York, NY 10029 USAEstrada, Y.论文数: 0 引用数: 0 h-index: 0机构: Icahn Sch Med Mt Sinai, New York, NY 10029 USA Icahn Sch Med Mt Sinai, New York, NY 10029 USABanerjee, A.论文数: 0 引用数: 0 h-index: 0机构: Pfizer Inc, Cambridge, England Icahn Sch Med Mt Sinai, New York, NY 10029 USAZhang, W.论文数: 0 引用数: 0 h-index: 0机构: Pfizer Inc, Cambridge, England Icahn Sch Med Mt Sinai, New York, NY 10029 USAZhu, L.论文数: 0 引用数: 0 h-index: 0机构: Pfizer Inc, Cambridge, England Icahn Sch Med Mt Sinai, New York, NY 10029 USABanfield, C.论文数: 0 引用数: 0 h-index: 0机构: Pfizer Inc, Cambridge, England Icahn Sch Med Mt Sinai, New York, NY 10029 USACox, L.论文数: 0 引用数: 0 h-index: 0机构: Pfizer Inc, Cambridge, England Icahn Sch Med Mt Sinai, New York, NY 10029 USAVincent, M.论文数: 0 引用数: 0 h-index: 0机构: Pfizer Inc, Cambridge, England Icahn Sch Med Mt Sinai, New York, NY 10029 USAPeeva, E.论文数: 0 引用数: 0 h-index: 0机构: Pfizer Inc, Cambridge, England Icahn Sch Med Mt Sinai, New York, NY 10029 USA
- [5] Safety of the oral JAK3/TEC inhibitor ritlecitinib (PF-06651600) in patients with alopecia areata: Results from the ALLEGRO phase 2b/3, randomized, double-blind, placebo-controlled trialJOURNAL OF THE AMERICAN ACADEMY OF DERMATOLOGY, 2022, 87 (03) : AB106 - AB106King, Brett论文数: 0 引用数: 0 h-index: 0机构: Yale Sch Med, New Haven, CT USA Yale Sch Med, New Haven, CT USASzepietowski, Jacek C.论文数: 0 引用数: 0 h-index: 0机构: Wroclaw Med Univ, Dept Dermatol Venereol & Allergol, Wroclaw, Poland Yale Sch Med, New Haven, CT USAFarrant, Paul论文数: 0 引用数: 0 h-index: 0机构: Univ Hosp Sussex, Dept Dermatol, Brighton Gen Hosp, Brighton, E Sussex, England Yale Sch Med, New Haven, CT USA
- [6] Efficacy of the oral JAK3/TEC inhibitor ritlecitinib (PF-06651600) in patients with alopecia areata over 48 weeks: Results from the ALLEGRO Phase 2b/3 randomized, double-blind, placebocontrolled trialJOURNAL OF THE AMERICAN ACADEMY OF DERMATOLOGY, 2022, 87 (03) : AB54 - AB54Mesinkovska, Natasha论文数: 0 引用数: 0 h-index: 0机构: Univ Calif Irvine, Sch Med, Irvine, CA 92717 USA Univ Calif Irvine, Sch Med, Irvine, CA 92717 USAShapiro, Jerry论文数: 0 引用数: 0 h-index: 0机构: NYU, Sch Med, New York, NY USA Univ Calif Irvine, Sch Med, Irvine, CA 92717 USAKing, Brett论文数: 0 引用数: 0 h-index: 0机构: Yale Univ, Sch Med, New Haven, CT USA Univ Calif Irvine, Sch Med, Irvine, CA 92717 USA
- [7] Design of a Janus Kinase 3 (JAK3) Specific Inhibitor 1-(2s,5R)-5-((7H-Pyrrolo[2,3-d]pyrimidin-4-yl)amino)-2-methylpiperidin-1-y1)prop-2-en-1-one (PF-06651600) Allowing for the Interrogation of JAK3 Signaling in HumansJOURNAL OF MEDICINAL CHEMISTRY, 2017, 60 (05) : 1971 - 1993Thorarensen, Atli论文数: 0 引用数: 0 h-index: 0机构: Pfizer Worldwide R&D, Worldwide Med Chem, 610 Main St, Cambridge, MA 02139 USA Pfizer Worldwide R&D, Worldwide Med Chem, 610 Main St, Cambridge, MA 02139 USADowty, Martin E.论文数: 0 引用数: 0 h-index: 0机构: Pfizer Worldwide R&D, Pharmacokinet Dynam & Metab, 1 Burtt Rd, Andover, MA 01810 USA Pfizer Worldwide R&D, Pharmacokinet Dynam & Metab, Eastern Point Rd, Groton, CT 06340 USA Pfizer Worldwide R&D, Worldwide Med Chem, 610 Main St, Cambridge, MA 02139 USABanker, Mary Ellen论文数: 0 引用数: 0 h-index: 0机构: Pfizer Worldwide R&D, Primary Pharmacol Grp, Eastern Point Rd, Groton, CT 06340 USA Pfizer Worldwide R&D, Worldwide Med Chem, 610 Main St, Cambridge, MA 02139 USAJuba, Brian论文数: 0 引用数: 0 h-index: 0机构: Pfizer Worldwide R&D, Inflammat & Immunol, 610 Main St, Cambridge, MA 02139 USA Pfizer Worldwide R&D, Worldwide Med Chem, 610 Main St, Cambridge, MA 02139 USAJussif, Jason论文数: 0 引用数: 0 h-index: 0机构: Pfizer Worldwide R&D, Inflammat & Immunol, 610 Main St, Cambridge, MA 02139 USA Pfizer Worldwide R&D, Worldwide Med Chem, 610 Main St, Cambridge, MA 02139 USALin, Tsung论文数: 0 引用数: 0 h-index: 0机构: Pfizer Worldwide R&D, Inflammat & Immunol, 610 Main St, Cambridge, MA 02139 USA Pfizer Worldwide R&D, Worldwide Med Chem, 610 Main St, Cambridge, MA 02139 USAVincent, Fabien论文数: 0 引用数: 0 h-index: 0机构: Pfizer Worldwide R&D, Primary Pharmacol Grp, Eastern Point Rd, Groton, CT 06340 USA Pfizer Worldwide R&D, Worldwide Med Chem, 610 Main St, Cambridge, MA 02139 USACzerwinski, Robert M.论文数: 0 引用数: 0 h-index: 0机构: Pfizer Worldwide R&D, Inflammat & Immunol, 610 Main St, Cambridge, MA 02139 USA Pfizer Worldwide R&D, Worldwide Med Chem, 610 Main St, Cambridge, MA 02139 USACasimiro-Garcia, Agustin论文数: 0 引用数: 0 h-index: 0机构: Pfizer Worldwide R&D, Worldwide Med Chem, 610 Main St, Cambridge, MA 02139 USA Pfizer Worldwide R&D, Worldwide Med Chem, 610 Main St, Cambridge, MA 02139 USAUnwalla, Ray论文数: 0 引用数: 0 h-index: 0机构: Pfizer Worldwide R&D, Worldwide Med Chem, 610 Main St, Cambridge, MA 02139 USA Pfizer Worldwide R&D, Worldwide Med Chem, 610 Main St, Cambridge, MA 02139 USATrujillo, John I.论文数: 0 引用数: 0 h-index: 0机构: Pfizer Worldwide R&D, Worldwide Med Chem, Eastern Point Rd, Groton, CT 06340 USA Pfizer Worldwide R&D, Worldwide Med Chem, 610 Main St, Cambridge, MA 02139 USALiang, Sidney论文数: 0 引用数: 0 h-index: 0机构: Pfizer Worldwide R&D, Worldwide Med Chem, Eastern Point Rd, Groton, CT 06340 USA Pfizer Worldwide R&D, Worldwide Med Chem, 610 Main St, Cambridge, MA 02139 USABalbo, Paul论文数: 0 引用数: 0 h-index: 0机构: Pfizer Worldwide R&D, Inflammat & Immunol, 610 Main St, Cambridge, MA 02139 USA Pfizer Worldwide R&D, Worldwide Med Chem, 610 Main St, Cambridge, MA 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- [8] Dual Inhibition of TYK2 and JAK1 for the Treatment of Autoimmune Diseases: Discovery of ((S)-2,2-Difluorocyclopropyl)((1R,5S)-3-(2-(1-methyl-1H-pyrazol-4-yl)amino)pyrimidin-4-yl)-3,8-diazabicyclo[3.2.1]octan-8-yl)methanone (PF-06700841)JOURNAL OF MEDICINAL CHEMISTRY, 2018, 61 (19) : 8597 - 8612Fensome, Andrew论文数: 0 引用数: 0 h-index: 0机构: Pfizer Inc, Med Design, 1 Portland St, Cambridge, MA 02139 USA Pfizer Inc, Med Design, 1 Portland St, Cambridge, MA 02139 USAAmbler, Catherine M.论文数: 0 引用数: 0 h-index: 0机构: Pfizer Inc, Med Design, Eastern Point Rd, Groton, CT 06340 USA Pfizer Inc, Med Design, 1 Portland St, Cambridge, MA 02139 USAArnold, Eric论文数: 0 引用数: 0 h-index: 0机构: Pfizer Inc, Med Design, Eastern Point Rd, Groton, CT 06340 USA Pfizer Inc, Med Design, 1 Portland St, Cambridge, MA 02139 USABanker, Mary Ellen论文数: 0 引用数: 0 h-index: 0机构: Pfizer Inc, Med Design, Eastern Point Rd, Groton, CT 06340 USA Pfizer Inc, Med Design, 1 Portland St, Cambridge, MA 02139 USABrown, Matthew F.论文数: 0 引用数: 0 h-index: 0机构: Pfizer Inc, Med Design, Eastern Point Rd, Groton, CT 06340 USA Pfizer Inc, Med Design, 1 Portland St, Cambridge, MA 02139 USAChrencik, Jill论文数: 0 引用数: 0 h-index: 0机构: Pfizer Inc, Med Design, Eastern Point Rd, Groton, CT 06340 USA Pfizer Inc, Med Design, 1 Portland St, Cambridge, MA 02139 USAClark, James D.论文数: 0 引用数: 0 h-index: 0机构: Pfizer Inc, Inflammat & Immunol, 1 Portland St, Cambridge, MA 02139 USA Pfizer Inc, Med Design, 1 Portland St, Cambridge, MA 02139 USADowty, Martin E.论文数: 0 引用数: 0 h-index: 0机构: Pfizer Inc, Med Design, 1 Portland St, Cambridge, MA 02139 USA Pfizer Inc, Med Design, 1 Portland St, Cambridge, MA 02139 USAEfremov, Ivan V.论文数: 0 引用数: 0 h-index: 0机构: Pfizer Inc, Med Design, 1 Portland St, Cambridge, MA 02139 USA Pfizer Inc, Med Design, 1 Portland St, Cambridge, MA 02139 USAFlick, Andrew论文数: 0 引用数: 0 h-index: 0机构: Pfizer Inc, Med Design, Eastern Point Rd, Groton, CT 06340 USA Pfizer Inc, Med Design, 1 Portland St, Cambridge, MA 02139 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