Multicomponent Reactions for the Synthesis of Functionalized Imidazoles

被引：5

作者：

Seyfi, Samereh ^{[1
]}

Hossaini, Zinatossadat ^{[1
]}

Rostami-Charati, Faramarz ^{[2
]}

机构：

[1] Islamic Azad Univ, Dept Chem, Qaemshahr Branch, Qaemshahr, Iran

[2] Gonbad Kavous Univ, Fac Sci, Dept Chem, Gonbad, Iran

来源：

COMBINATORIAL CHEMISTRY & HIGH THROUGHPUT SCREENING | 2013年 / 16卷 / 08期

关键词：

Arylisothiocyanates; dialkyl acetylenedicarboxylates; multi component reaction; ninhydrin; primary amine; CHEMISTRY;

D O I：

10.2174/13862073113169990005

中图分类号：

Q5 [生物化学];

学科分类号：

071010 ; 081704 ;

摘要：

An efficient synthesis of functionalized tetrahydroimidazoles via a one-pot tandem reaction between ninhydrin, primary alkylamines, arylisocyanates or arylisothiocyanates, acetylenic esters and triphenylphosphine is described.

引用

页码：652 / 656

页数：5

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