Development of a new 18F-labeled radioligand for imaging sigma2 receptors by positron emission tomography

被引:0
作者
Ludwig, Friedrich-Alexander [1 ]
Fischer, Steffen [2 ]
Moldovan, Rares [3 ]
Deuther-Conrad, Winnie
Kranz, Mathias
Schepmann, Dirk [4 ]
Jia, Hongmei [5 ]
Wunsch, Bernhard
Brust, Peter [6 ]
机构
[1] Helmholtz Zentrum Dresden Rossendorf, Dept Neuroradiopharmaceut, Inst Radiopharmaceut Canc Res, Res Site Leipzig, Dresden, Germany
[2] HZDR, FS Leipzig, Dresden, Germany
[3] Helmholtz Zentrum Dresden Rossendorf, Inst Radiopharmaceut Canc Res, Dresden, Germany
[4] Univ Munster, Dept Pharmaceut & Med Chem, Munster, Germany
[5] Beijing Normal Univ, Beijing, Peoples R China
[6] Helmholtz Zentrum Dresden Rossendorf, Dresden, Germany
关键词
D O I
暂无
中图分类号
Q5 [生物化学];
学科分类号
071010 ; 081704 ;
摘要
P-027
引用
收藏
页码:S181 / S182
页数:2
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[1]   Sigma Receptor (σR) Ligands with Antiproliferative and Anticancer Activity [J].
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MOLECULES, 2017, 22 (09)
[2]   18F-Labeled indole-based analogs as highly selective radioligands for imaging sigma-2 receptors in the brain [J].
Wang, Liang ;
Ye, Jiajun ;
He, Yingfang ;
Deuther-Conrad, Winnie ;
Zhang, Jinming ;
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Steinbach, Joerg ;
Huang, Yiyun ;
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Jia, Hongmei .
BIOORGANIC & MEDICINAL CHEMISTRY, 2017, 25 (14) :3792-3802