F 11356, a novel 5HT derivative with unique high intrinsic activity at 5HT1B/1D receptors in models relevant to migraine.

被引:0
作者
John, GW [1 ]
Pauwels, PJ [1 ]
Perez, M [1 ]
Halazy, S [1 ]
Le Grand, B [1 ]
Verscheure, Y [1 ]
Valentin, JP [1 ]
Palmier, C [1 ]
Wurch, T [1 ]
Chopin, P [1 ]
Marien, M [1 ]
Colpaert, FC [1 ]
机构
[1] Ctr Rech Pierre Fabre, F-81106 Castres, France
关键词
D O I
暂无
中图分类号
R74 [神经病学与精神病学];
学科分类号
摘要
引用
收藏
页码:404 / 404
页数:1
相关论文
共 50 条
[31]   Serotonin inhibits trigeminal nucleus activity evoked by craniovascular stimulation through a 5HT1B/1D receptor:: A central action in migraine? [J].
Goadsby, PJ ;
Hoskin, KL .
ANNALS OF NEUROLOGY, 1998, 43 (06) :711-718
[32]   THE ROLE OF PERIPHERAL 5-HT1A, 5-HT1B, 5-HT1D, 5-HT1E AND 5-HT1F SEROTONERGIC RECEPTORS IN THE REDUCTION OF NOCICEPTION IN RATS [J].
Granados-Soto, V. ;
Arguelles, C. F. ;
Rocha-Gonzalez, H. I. ;
Godinez-Chaparro, B. ;
Flores-Murrieta, F. J. ;
Villalon, C. M. .
NEUROSCIENCE, 2010, 165 (02) :561-568
[33]   In vivo pharmacological actions of F 11356, a novel high efficacy anti-migraine 5-HT1B/D receptor agonist. [J].
John, GW ;
Verscheure, Y ;
Infanti, F ;
Bel, L ;
Perez, M ;
Halazy, S ;
Chopin, P ;
Marien, M ;
Colpaert, FC .
NAUNYN-SCHMIEDEBERGS ARCHIVES OF PHARMACOLOGY, 1998, 358 (01) :R523-R523
[34]   Frovatriptan succinate, a 5-HT1B/1D receptor agonist for migraine [J].
Balbisi, EA .
INTERNATIONAL JOURNAL OF CLINICAL PRACTICE, 2004, 58 (07) :695-705
[35]   Do 5HT1B/1D receptor agonists have an effect on mood and anxiety disorders? [J].
Morelli, Nicola ;
Gori, Sara ;
Choub, Anna ;
Maluccio, Maria Rosaria ;
Orlandi, Giovanni ;
Guazzelli, Mario ;
Murri, Luigi .
CEPHALALGIA, 2007, 27 (05) :471-472
[36]   RU24969 induced behavioural syndrome requires activation of both 5HT(1A) and 5HT(1B) receptors [J].
ONeill, MF ;
Parameswaran, T .
PSYCHOPHARMACOLOGY, 1997, 132 (03) :255-260
[37]   5HT1A and 5HT1B receptors of medial prefrontal cortex modulate anxiogenic-like behaviors in rats [J].
Solati, Jalal ;
Salari, Ali-Akbar ;
Bakhtiari, Amir .
NEUROSCIENCE LETTERS, 2011, 504 (03) :325-329
[38]   INTERACTION OF THE ALPHA-ADRENOCEPTOR AGONIST OXYMETAZOLINE WITH SEROTONIN 5-HT1A-RECEPTORS, 5-HT1B-RECEPTORS, 5-HT1C-RECEPTORS AND 5-HT1D-RECEPTORS [J].
SCHOEFFTER, P ;
HOYER, D .
EUROPEAN JOURNAL OF PHARMACOLOGY, 1991, 196 (02) :213-216
[39]   5-HT1A and 5-HT1B/1D receptors are involved in the modulation of the trigeminovascular system of the cat:: a microiontophoretic study [J].
Boers, PM ;
Donaldson, C ;
Zagami, AS ;
Lambert, GA .
NEUROPHARMACOLOGY, 2000, 39 (10) :1833-1847
[40]   SAR study on close analogs of F 11356:: A novel series of highly efficacious and selective H5HT1B/1D receptor agonists for the acute treatment of migraine [J].
Perez, M ;
Pallard, I ;
Fourrier, C ;
Potier, P ;
Pauwels, PJ ;
Vaientin, JF ;
John, GW ;
Halazy, S .
ABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY, 1998, 216 :U244-U244